133 results on '"Brimble, Margaret"'
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2. Analysis of Advanced Glycation End products in ribose-, glucose- and lactose-crosslinked gelatin to correlate the physical changes induced by Maillard reaction in films
3. C-2 derivatized 8-sulfonamidoquinolines as antibacterial compounds
4. Synthetic approaches towards bedaquiline and its derivatives
5. Naturally occurring antitubercular cyclic peptides
6. Natural product derived privileged scaffolds in drug discovery
7. Synthesis and antiproliferative activity of culicinin D analogues containing simplified AHMOD-based residues
8. Anthranilate phosphoribosyltransferase: Binding determinants for 5′-phospho-alpha-d-ribosyl-1′-pyrophosphate (PRPP) and the implications for inhibitor design
9. Structure-activity relationship study of the tumour-targeting peptide A20FMDV2 via modification of Lys16, Leu13, and N- and/or C-terminal functionality
10. Multifunctional thermoresponsive designer peptide hydrogels
11. Controlling gelation with sequence: Towards programmable peptide hydrogels
12. Synthesis and biological evaluation of analogues of the potent ADAM8 inhibitor cyclo(RLsKDK) for the treatment of inflammatory diseases and cancer metastasis
13. Stereoselective synthesis of the rat selective toxicant norbormide
14. Identification of anticancer agents based on the thieno[2,3-b]pyridine and 1H-pyrazole molecular scaffolds
15. Enantioselective synthesis of BE ring analogues of methyllycaconitine
16. Electrochemically-controlled grafting of hydrophilic brushes from conducting polymer substrates
17. Formal synthesis of nanaomycin D via a Hauser–Kraus annulation using a chiral enone-lactone
18. Regulation and Quality Control of Adiponectin Assembly by Endoplasmic Reticulum Chaperone ERp44
19. A review of the synthesis of α-carbolines
20. Glucose as an agent of post-translational modification in diabetes — New cardiac epigenetic insights
21. Studies towards development of asymmetric double-Mannich reactions of chiral 2-oxocyclohexanecarboxylate derivatives with bis(aminol)ethers
22. Synthesis of the carbon skeleton of the griseorhodins
23. Synthesis and evaluation of 9-deoxy analogues of (−)-thysanone, an inhibitor of HRV 3C protease
24. Synthesis and biological evaluation of the osteoblast proliferating cyclic peptides dianthins G and H
25. Synthesis of truncated analogues of preptin-(1–16), and investigation of their ability to stimulate osteoblast proliferation
26. Synthesis and methemoglobinemia-inducing properties of benzocaine isosteres designed as humane rodenticides
27. Synthesis of highly substituted pyranonaphthalene spiroketals related to the griseusins using a Hauser–Kraus annulation strategy
28. Synthesis of the spiroacetal core of the cephalosporolide family of natural products
29. Synthesis and cytotoxicity of pyranonaphthoquinone natural product analogues under bioreductive conditions
30. Prodrugs of N-dicarboximide derivatives of the rat selective toxicant norbormide
31. Structure and dynamics of human Nedd4-1 WW3 in complex with the αENaC PY motif
32. A new precursor for conducting polymer-based brush interfaces with electroactivity in aqueous solution
33. DNA adduct formation of mitomycin C. A test case for DFT calculations on model systems
34. How to blast osteoblasts? Novel dicarba analogues of amylin-(1–8) to treat osteoporosis
35. Synthesis and biological evaluation of tyrosine modified analogues of the α4β7 integrin inhibitor biotin-R8ERY
36. Access to 2-alkyl chromanones via a conjugate addition approach
37. A tandem Diels–Alder/Mannich approach to the synthesis of AE and ABE ring analogues of Delphinium alkaloids
38. Design and synthesis of prodrugs of the rat selective toxicant norbormide
39. Tyrosine modified analogues of the α4β7 integrin inhibitor biotin-R8ERY prepared via Click Chemistry: Synthesis and biological evaluation
40. Synthesis and evaluation of disulfide bond mimetics of amylin-(1–8) as agents to treat osteoporosis
41. An efficient synthesis of 3-alkyl-1,5,3-dioxazepanes and their use as electrophiles in double-Mannich reactions
42. The enantioselective synthesis of tetracyclic methyllycaconitine analogues
43. Influence of α-methyl substitution of proline-based organocatalysts on the asymmetric α-oxidation of aldehydes
44. Pyranonaphthoquinone derivatives of eleutherin, ventiloquinone L, thysanone and nanaomycin A possessing a diverse topoisomerase II inhibition and cytotoxicity spectrum
45. In vitro metabolism of norbormide in rat, mouse and guinea pig liver preparations
46. NNZ-2566: A Gly–Pro–Glu analogue with neuroprotective efficacy in a rat model of acute focal stroke
47. Anti- Helicobacter pylori activity of derivatives of the phthalide-containing antibacterial agents spirolaxine methyl ether, CJ-12,954, CJ-13,013, CJ-13,102, CJ-13,104, CJ-13,108 and CJ-13,015
48. Chemoenzymatic synthesis of deoxy analogues of the DNA topoisomerase II inhibitor eleutherin and the 3C-protease inhibitor thysanone
49. An approach to an enantioselective synthesis of crisamicin A via a novel double Hauser–Kraus annulation strategy
50. Synthesis of a C8 oxygenated pyranonaphthoquinone: a useful precursor to dimeric pyranonaphthoquinones
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