25 results on '"Keith, John"'
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2. The SAR of brain penetration for a series of heteroaryl urea FAAH inhibitors
3. Understanding DP receptor antagonism using a CoMSIA approach
4. Synthesis of 7-chloro-2,3-dihydro-2-[1-(pyridinyl)alkyl]-pyridazino[4,5- b ]quinoline-1,4,10(5 H )-triones as NMDA glycine-site antagonists
5. 1-Aryl-2-((6-aryl)pyrimidin-4-yl)amino)ethanols as competitive inhibitors of fatty acid amide hydrolase
6. Heteroarylureas with spirocyclic diamine cores as inhibitors of fatty acid amide hydrolase
7. Heteroaryl urea inhibitors of fatty acid amide hydrolase: Structure–mutagenicity relationships for arylamine metabolites
8. Pre-clinical characterization of aryloxypyridine amides as histamine H3 receptor antagonists: Identification of candidates for clinical development
9. Thiadiazolopiperazinyl ureas as inhibitors of fatty acid amide hydrolase
10. 2-Aryloxymethylmorpholine histamine H 3 antagonists
11. Synthesis and biological activity of piperazine and diazepane amides that are histamine H 3 antagonists and serotonin reuptake inhibitors
12. Dual serotonin transporter inhibitor/histamine H 3 antagonists: Development of rigidified H 3 pharmacophores
13. Pyrrolidino-tetrahydroisoquinolines bearing pendant heterocycles as potent dual H 3 antagonist and serotonin transporter inhibitors
14. Novel naphthyridines are histamine H 3 antagonists and serotonin reuptake transporter inhibitors
15. Pyrrolidino-tetrahydroisoquinolines as potent dual H 3 antagonist and serotonin transporter inhibitors
16. Novel tetrahydroisoquinolines are histamine H 3 antagonists and serotonin reuptake inhibitors
17. Dual serotonin transporter/histamine H 3 ligands: Optimization of the H 3 pharmacophore
18. 2-Aryloxymethylmorpholine histamine H3 antagonists
19. Synthesis and biological activity of piperazine and diazepane amides that are histamine H3 antagonists and serotonin reuptake inhibitors
20. Dual serotonin transporter inhibitor/histamine H3 antagonists: Development of rigidified H3 pharmacophores
21. Pyrrolidino-tetrahydroisoquinolines bearing pendant heterocycles as potent dual H3 antagonist and serotonin transporter inhibitors
22. Novel naphthyridines are histamine H3 antagonists and serotonin reuptake transporter inhibitors
23. Pyrrolidino-tetrahydroisoquinolines as potent dual H3 antagonist and serotonin transporter inhibitors
24. Dual serotonin transporter/histamine H3 ligands: Optimization of the H3 pharmacophore
25. Novel tetrahydroisoquinolines are histamine H3 antagonists and serotonin reuptake inhibitors
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