15 results on '"Xu, Yechun"'
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2. Drug repurposing and structure-based discovery of new PDE4 and PDE5 inhibitors
3. Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
4. Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2
5. In silico screening-based discovery of novel covalent inhibitors of the SARS-CoV-2 3CL protease
6. Design, synthesis, and biological evaluation of tetrahydroisoquinolines derivatives as novel, selective PDE4 inhibitors for antipsoriasis treatment
7. Structure-based design of potent FABP4 inhibitors with high selectivity against FABP3
8. Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors
9. Discovery, optimization and biological evaluation for novel c-Met kinase inhibitors
10. Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor
11. Novel fatty acid binding protein 4 (FABP4) inhibitors: Virtual screening, synthesis and crystal structure determination
12. Discovery of potent N-(isoxazol-5-yl)amides as HSP90 inhibitors
13. Discovery of pyrazole as C-terminus of selective BACE1 inhibitors
14. Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3- b ][1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor
15. Discovery, optimization and biological evaluation for novel c-Met kinase inhibitors.
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