43 results on '"Fedorov, Oleg"'
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2. Discovery of a Potent, Selective, and Cell-Active SPIN1 Inhibitor
3. Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist.
4. Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist
5. Discovery of High-Affinity Small-Molecule Binders of the Epigenetic Reader YEATS4
6. Discovery of High-Affinity Small-Molecule Binders of the Epigenetic Reader YEATS4.
7. Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold
8. Discovery and Characterization of Selective and Ligand-Efficient DYRK Inhibitors
9. Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain
10. DFG-1 Residue Controls Inhibitor Binding Mode and Affinity, Providing a Basis for Rational Design of Kinase Inhibitor Selectivity
11. 8-substituted pyrido[3,4-d]pyrimidin-4(3H)-one derivatives as potent, cell permeable, KDM4 (JMJD2) and KDM5 (JARID1) histone lysine demethylase inhibitors
12. A Chemical Probe for Tudor Domain Protein Spindlin1 to Investigate Chromatin Function
13. Discovery of a Potent and Selective Fragment-like Inhibitor of Methyllysine Reader Protein Spindlin 1 (SPIN1)
14. SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK)
15. Structure Enabled Design of BAZ2-ICR, A Chemical Probe Targeting the Bromodomains of BAZ2A and BAZ2B
16. Structure-Based Approach toward Identification of Inhibitory Fragments for Eleven-Nineteen-Leukemia Protein (ENL)
17. Creation of a Novel Class of Potent and Selective MutT Homologue 1 (MTH1) Inhibitors Using Fragment-Based Screening and Structure-Based Drug Design
18. Design of a Chemical Probe for the Bromodomain and Plant Homeodomain Finger-Containing (BRPF) Family of Proteins
19. Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains
20. Design of a Biased Potent Small Molecule Inhibitor of the Bromodomain and PHD Finger-Containing (BRPF) Proteins Suitable for Cellular and in Vivo Studies
21. Development of Selective CBP/P300 Benzoxazepine Bromodomain Inhibitors
22. Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis
23. Identification and Development of 2,3-Dihydropyrrolo[1,2-a]quinazolin-5(1H)-one Inhibitors Targeting Bromodomains within the Switch/Sucrose Nonfermenting Complex
24. Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
25. Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor
26. Structure-Based Identification of Inhibitory Fragments Targeting the p300/CBP-Associated Factor Bromodomain
27. Discovery of novel small-molecule inhibitors of BRD4 using structure-based virtual screening
28. Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF
29. Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B
30. [1,2,4]Triazolo[4,3-a]phthalazines: Inhibitors of Diverse Bromodomains
31. Targeting Low-Druggability Bromodomains: Fragment Based Screening and Inhibitor Design against the BAZ2B Bromodomain
32. Optimization of 3,5-Dimethylisoxazole Derivatives as Potent Bromodomain Ligands
33. Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF.
34. Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B.
35. 7,8-Dichloro-1-oxo-β-carbolines as a Versatile Scaffold for the Development of Potent and Selective Kinase Inhibitors with Unusual Binding Modes
36. 3,5-Dimethylisoxazoles Act As Acetyl-lysine-mimetic Bromodomain Ligands
37. Leucettines, a Class of Potent Inhibitors of cdc2-Like Kinases and Dual Specificity, Tyrosine Phosphorylation Regulated Kinases Derived from the Marine Sponge Leucettamine B: Modulation of Alternative Pre-RNA Splicing
38. Structural Basis of Inhibitor Specificity of the Human Protooncogene Proviral Insertion Site in Moloney Murine Leukemia Virus (PIM-1) Kinase
39. [1,2,4]Triazolo[4,3-a]phthalazines:Inhibitors of Diverse Bromodomains.
40. Targeting Low-DruggabilityBromodomains: FragmentBased Screening and Inhibitor Design against the BAZ2B Bromodomain.
41. Discovery of Novel Small-MoleculeInhibitors of BRD4Using Structure-Based Virtual Screening.
42. Optimizationof 3,5-Dimethylisoxazole Derivativesas Potent Bromodomain Ligands.
43. Discovery and Characterization of GSK2801, a Selective Chemical Probe for the Bromodomains BAZ2A and BAZ2B.
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