31 results on '"van der Stelt, Mario"'
Search Results
2. Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
3. Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D
4. Structure–Activity Relationship Studies of α-Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family
5. Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors
6. Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N‑Acylphosphatidylethanolamine Phospholipase D.
7. Activity-Based Protein Profiling Delivers Selective Drug Candidate ABX-1431, a Monoacylglycerol Lipase Inhibitor, To Control Lipid Metabolism in Neurological Disorders
8. An Affinity-Based Probe for the Human Adenosine A2A Receptor
9. Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding
10. Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors
11. Structure-Based Design of β5c Selective Inhibitors of Human Constitutive Proteasomes
12. Comprehensive Analysis of Structure–Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α Inhibitors
13. An Affinity-Based Probe for the Human Adenosine A2A Receptor.
14. Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding.
15. Identification and Development of Biphenyl Substituted Iminosugars as Improved Dual Glucosylceramide Synthase/Neutral Glucosylceramidase Inhibitors
16. N-Tetradecylcarbamyl Lipopeptides as Novel Agonists for Toll-like Receptor 2
17. Discovery of Glycine Sulfonamides as Dual Inhibitors of sn-1-Diacylglycerol Lipase α and α/β-Hydrolase Domain 6
18. Structure-Based Design of β1i or β5i Specific Inhibitors of Human Immunoproteasomes
19. Incorporation of Non-natural Amino Acids Improves Cell Permeability and Potency of Specific Inhibitors of Proteasome Trypsin-like Sites
20. Comprehensive Analysis of Structure-Activity Relationships of a-Ketoheterocycles as sn-1-Diacylglycerol Lipase a Inhibitors.
21. Discovery and Optimization of 1-(4-(Pyridin-2-yl)benzyl)imidazolidine-2,4-dione Derivatives As a Novel Class of Selective Cannabinoid CB2 Receptor Agonists
22. Identification and Developmentof Biphenyl SubstitutedIminosugars as Improved Dual Glucosylceramide Synthase/Neutral GlucosylceramidaseInhibitors.
23. Oxygenated Metabolites of Anandamide and 2-Arachidonoylglycerol: Conformational Analysis and Interaction with Cannabinoid Receptors, Membrane Transporter, and Fatty Acid Amide Hydrolase
24. N-Tetradecylcarbamyl Lipopeptidesas Novel Agonists for Toll-like Receptor 2.
25. Discovery of Glycine Sulfonamidesas Dual Inhibitorsof sn-1-Diacylglycerol Lipase α and α/β-HydrolaseDomain 6.
26. Structure-Based Design ofβ1i or β5i SpecificInhibitors of Human Immunoproteasomes.
27. Incorporation of Non-naturalAmino Acids ImprovesCell Permeability and Potency of Specific Inhibitors of ProteasomeTrypsin-like Sites.
28. Structure-Based Design of β5c Selective Inhibitors of Human Constitutive Proteasomes.
29. Structure-Guided Discovery of cis -Hexahydro-pyrido-oxazinones as Reversible, Drug-like Monoacylglycerol Lipase Inhibitors.
30. An Affinity-Based Probe for the Human Adenosine A 2A Receptor.
31. Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding.
Catalog
Books, media, physical & digital resources
Discovery Service for Jio Institute Digital Library
For full access to our library's resources, please sign in.