92 results on '"Jarvest, Richard L."'
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2. 6-Alkylquinolone-3-carboxylic acid tethered to macrolides synthesis and antimicrobial profile
3. New atropisomeric biaryl derivatives of 4-aminopyridine—identification of an improved nucleophilic catalyst for asymmetric acylation of sec-alcohols
4. Interaction of tyrosyl aryl dipeptides with S. aureus tyrosyl tRNA synthetase: Inhibition and crystal structure of a complex
5. Inhibition of human cytomegalovirus protease by enedione derivatives of thieno[2,3-d]oxazinones through a novel dual acylation/alkylation mechanism
6. Inhibition of herpes proteases and antiviral activity of 2-substituted thieno[2,3-d]oxazinones
7. Concise, synthesis, preparation resolution, absolute configuration determination, and applications of an atropisomeric biaryl catalysts for asymmetric acylation
8. Synthesis and antiviral activity of novel HCV NS3 protease inhibitors with P4 capping groups
9. Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties
10. Synthesis and evaluation of novel α-amino cyclic boronates as inhibitors of HCV NS3 protease
11. Novel macrocyclic HCV NS3 protease inhibitors derived from α-amino cyclic boronates
12. Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 protease
13. Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 protease
14. Discovery and optimisation of potent, selective, ethanolamine inhibitors of bacterial phenylalanyl tRNA synthetase
15. Definition of the heterocyclic pharmacophore of bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues
16. Discovery of Novel Urea-Based Hepatitis C Protease Inhibitors with High Potency against Protease-Inhibitor-Resistant Mutants.
17. Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-Positive antibacterial activity
18. Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity
19. Concise Synthesis, Preparative Resolution, Absolute Configuration Determination, and Applications, and Applications of an Atropisomeric Biaryl Catalyst for Asymmetric Acylation.
20. Crystal structure of Staphylococcus aureus tyrosyl-tRNA synthetase in complex with a class of potent and specific inhibitors.
21. The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase
22. Potent synthetic inhibitors of tyrosyl tRNA synthetase derived from C-pyranosyl analogues of SB-219383
23. Synthetic analogues of SB-219383. Novel C-glycosyl peptides as inhibitors of tyrosyl tRNA synthetase
24. Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Carbocyclic Analogues of the Natural Product SB-219383
25. A stereochemical investigation of the cyclisation of D-glucose-6[(R)-16O,17O,18O]phosphate and adenosine-5′[(R)-16O,17O,18O]phosphate.
26. Crystal and Molecular Structures of the Antiviral Acyclonucleoside 9-[4-Hydroxy-3-(hydroxymethyl)butyl]guanine (BRL 39123, Penciclovir) and its Prodrug 9-[4-Acetoxy-3-(acetoxymethyl)butyl]-2-aminopurine (BRL 42810, Famciclovir).
27. Exploring the active site of herpes simplex virus type-1 thymidine kinase by X-ray crystallography of complexes with aciclovir and other ligands.
28. Analysis of the chirality of [16O,17O,18O] phosphate esters by 31P nuclear magnetic resonance spectroscopy.
29. Synthesis of [3-(phosphonomethoxy)pyrrolidin-1-yl] derivatives of pyrimidines and purines: analogues of 2′,3′-dideoxynucleotides.
30. Chemoenzymatic approach to the synthesis of the antiviral agents penciclovir and famciclovir in isotopically chiral [13C] labelled form.
31. Pyrrolidine analogues of 2′,3′-dideoxynucleosides: synthesis via 9-aminopurines and 1-aminopyrimidines.
32. Analogues of the antiviral acyclonucleoside 9-(4-hydroxy-3-hydroxymethylbutyl)guanine. Part 4. Substitution on the 2-amino group.
33. Analogues of the antiviral acyclonucleoside 9-(4-hydroxy-3-hydroxymethylbutyl)guanine. Part 3. Modification of a 3′-hydroxymethyl group.
34. Aminoalkyl adenylate and aminoacyl sulfamate intermediate analogues differing greatly in affinity for their cognate Staphylococcus aureus aminoacyl tRNA synthetases
35. Inhibitors of bacterial tyrosyl tRNA synthetase: synthesis of four stereoisomeric analogues of the natural product SB-219383
36. The synthesis of 5-alkoxy and 5-amino substituted thiophenes
37. The stereochemical course of the hydrolysis of cyclic AMP by beef heart cyclic AMP phosphodiesterase.
38. Synthesis of methyl (R)- and (S)-[18O]phosphorothioates and determination of the absolute configuration at phosphorus of the diastereoisomers of adenosine 5′-(1-thiotriphosphate).
39. Synthesis of N-phenylpyrrole and pyrazole amidines and related diamines.
40. The stereochemistry of 2-substituted-2-oxo-4,5-diphenyl-1,3,2-dioxaphospholans and the related chiral [16O,17O,18O]phosphate monoesters.
41. Synthesis of isotopically chiral [13C]penciclovir (BRL 39123) and its use to determine the absolute configuration of penciclovir triphosphate formed in herpes virus infected cells.
42. Definition of the Heterocyclic Pharmacophore of Bacterial Methionyl tRNA Synthetase Inhibitors: Potent Antibacterially Active Non-quinolone Analogues.
43. New Atropisomeric Biaryl Derivatives of 4-Aminopyridine-Identification of an Improved Nucleophilic Catalyst for Asymmetric Acylation of sec-Alcohols.
44. Optimization of Aryl Substitution Leading to Potent Methionyl tRNA Synthetase Inhibitors with Excellent Gram-Positive Antibacterial Activity.
45. The Antimicrobial Natural Product Chuangxinmycin and Some Synthetic Analogues Are Potent and Selective Inhibitors of Bacterial Tryptophanyl tRNA Synthetase.
46. ChemInform Abstract: Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Carbocyclic Analogues of the Natural Product SB-219383.
47. ChemInform Abstract: Synthetic Analogues of SB-219383. Novel C-Glycosyl Peptides as Inhibitors of Tyrosyl tRNA Synthase.
48. ChemInform Abstract: Synthesis and Activity of Analogues of SB-219383: Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase.
49. ChemInform Abstract: Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Four Stereoisomeric Analogues of the Natural Product SB-219383.
50. ChemInform Abstract: Aminoalkyl Adenylate and Aminoacyl Sulfamate Intermediate Analogues Differing Greatly in Affinity for Their Cognate Staphylococcus aureus Aminoacyl tRNA Synthetases.
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