234 results on '"Csuk, Rene"'
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2. Disrupting protease and deubiquitinase activities of SARS-CoV-2 papain-like protease by natural and synthetic products discovered through multiple computational and biochemical approaches
3. Stereochemistry matters: Inhibition of carbonic anhydrase II by amino acid derived sulfamates depends on their absolute configuration
4. An asiatic acid derived trisulfamate acts as a nanomolar inhibitor of human carbonic anhydrase VA
5. Lupane acetates in small molecule drug hybrids: Probing their inhibitory activity for carbonic anhydrase II
6. Dehydroabietylamine derived bistetrazoles from ultrasound-assisted pseudo-seven-component Ugi reactions act as efficient and selective inhibitors of cholinesterases
7. Isosteviol – A new scaffold for the synthesis of carbonic anhydrase II inhibitors
8. Ready-to-use nanopore platform for label-free small molecule quantification: Ethanolamine as first example
9. Targeted theranostics: Near-infrared triterpenoic acid-rhodamine conjugates as prerequisites for precise cancer diagnosis and therapy
10. Triazole‐tethered boswellic acid derivatives against breast cancer: Synthesis, in vitro, and in‐silico studies
11. Non-cytotoxic aza-BODIPY triterpene conjugates to target the endoplasmic reticulum
12. Asiatic acid as a leading structure for derivatives combining sub-nanomolar cytotoxicity, high selectivity, and the ability to overcome drug resistance in human preclinical tumor models
13. Synthesis of novel substituted quinoline derivatives as diabetics II inhibitors and along with their in-silico studies
14. Synthesis and cytotoxicity of diastereomeric benzylamides derived from maslinic acid, augustic acid and bredemolic acid
15. On the influence of the rhodamine substituents onto the cytotoxicity of mitocanic maslinic acid rhodamine conjugates
16. New amides derived from sclareolide as anticholinesterase agents
17. Synthesis and antidepressant-like effects of new 5-epi-incensole and 5-epi- incensole acetate in chronic unpredictable mild stress model of depression; behavioural and biochemical correlates
18. Synthesis and cytotoxicity of apoptosis-inducing N-heterocyclic triterpene amides
19. An improved partial synthesis of corosolic acid and its conversion to highly cytotoxic mitocans
20. Incensole derivatives from frankincense: Isolation, enhancement, synthetic modification, and a plausible mechanism of their anti-depression activity
21. A tormentic acid-homopiperazine-rhodamine B conjugate of single-digit nanomolar cytotoxicity and high selectivity for several human tumor cell lines
22. Comparative study of the cytotoxicity, apoptotic, and epigenetic effects of Boswellic acid derivatives on breast cancer
23. Synthesis and structure of azelastine-N-oxides
24. Stable triterpenoid iminium salts and their activity as inhibitors of butyrylcholinesterase
25. Substrate-like novel inhibitors of prolyl specific oligo peptidase for neurodegenerative disorders.
26. N-methylated diazabicyclo[3.2.2]nonane substituted triterpenoic acids are excellent, hyperbolic and selective inhibitors for butyrylcholinesterase
27. Selective and low-cost triterpene urea and amide derivatives of high cytotoxicity and selectivity
28. A Malaprade cleavage, a McMurry ring closure and an intramolecular aldol contraction of maslinic acid’s ring A
29. Betulinic acid and glycyrrhetinic acid derived piperazinyl spacered rhodamine B conjugates are highly cytotoxic and necrotic
30. Hydroxyethylamide substituted triterpenoic acids hold good cytotoxicity for human tumor cells
31. Apoptotic activity of substituted 3-O-acetyl-betulinic acid benzylamides
32. MSBA-S – A pentacyclic sulfamate as a new option for radiotherapy of human breast cancer cells
33. Identification of new pharmacophore against SARS-CoV-2 spike protein by multi-fold computational and biochemical techniques
34. Cembranoids from Boswellia species
35. Biosynthetic diversity in triterpene cyclization within the Boswellia genus
36. Therapeutic potential of N4-substituted thiosemicarbazones as new urease inhibitors: Biochemical and in silico approach
37. Separating the true from the false: A rapid HPTLC-ESI-MS method for the determination of cannabinoids in different oils
38. Cytotoxic triterpenoid–safirinium conjugates target the endoplasmic reticulum
39. Betulinic acid derived amides are highly cytotoxic, apoptotic and selective
40. An unprecedented epimerization and annelation reaction of platanic acid amides
41. New amino acid clubbed Schiff bases inhibit carbonic anhydrase II, α-glucosidase, and urease enzymes: in silico and in vitro
42. Synthesis of some steroidal mitocans of nanomolar cytotoxicity acting by apoptosis
43. Synthesis and urease inhibitory activity of 1,4-benzodioxane-based thiosemicarbazones: Biochemical and computational approach
44. Synthesis and cytotoxic evaluation of hydroxycinnamic acid rhodamine B conjugates
45. Design, synthesis and cytotoxicity of BODIPY FL labelled triterpenoids
46. Toward more Sustainable Enzyme Reactions: Enhancing Kinetics by Polydimethylacrylamide Implementation
47. Ready-to-use nanopore platform for label-free small molecule quantification: Ethanolamine as first example
48. Evaluation of cholinesterase inhibitory activity and cytotoxicity of synthetic derivatives of di- and triterpene metabolites from Pinus silvestris and Dipterocarpus alatus resins
49. 2-O-(2-chlorobenzoyl) maslinic acid triggers apoptosis in A2780 human ovarian carcinoma cells
50. Caffeic acid phenethyl ester (CAPE)-derivatives act as selective inhibitors of acetylcholinesterase
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