398 results on '"van der Stelt, Mario"'
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2. A monoacylglycerol lipase inhibitor showing therapeutic efficacy in mice without central side effects or dependence
3. Structural basis of selective cannabinoid CB2 receptor activation
4. Dual allosteric and orthosteric pharmacology of synthetic analog cannabidiol-dimethylheptyl, but not cannabidiol, on the cannabinoid CB2 receptor
5. THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Enzymes
6. Multi-parameter optimization: Development of a morpholin-3-one derivative with an improved kinetic profile for imaging monoacylglycerol lipase in the brain
7. Oxygenation of Anandamide by Lipoxygenases
8. Fluorescence-Based NAPE-PLD Activity Assay
9. Cellular Assay to Study β-Arrestin Recruitment by the Cannabinoid Receptors 1 and 2
10. Semisynthetic guanidino lipoglycopeptides with potent in vitro and in vivo antibacterial activity.
11. P2X7 receptor‐dependent increase in endocannabinoid 2‐arachidonoyl glycerol production by neuronal cells in culture: Dynamics and mechanism.
12. Structure–Activity Relationship Studies of Aryl Sulfoxides as Reversible Monoacylglycerol Lipase Inhibitors.
13. Discovery of a Cannabinoid CB2 Receptor Fluorescent Probe Based on a Pyridin-2-yl-benzyl-imidazolidine-2,4-dione Scaffold.
14. Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
15. Stress-induced modulation of endocannabinoid signaling leads to delayed strengthening of synaptic connectivity in the amygdala
16. Discovery of a Photoaffinity Probe that Captures the Active Conformation of the Cannabinoid CB2 Receptor.
17. Opportunities for Lipid-Based Probes in the Field of Immunology
18. Biochemical and Cellular Characterization of the Function of Fluorophosphonate-Binding Hydrolase H (FphH) in Staphylococcus aureus Support a Role in Bacterial Stress Response
19. IMI European Lead Factory — democratizing access to high-throughput screening
20. PharmacoSTORM nanoscale pharmacology reveals cariprazine binding on Islands of Calleja granule cells
21. Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice
22. Improving CLL Vγ9Vδ2-T–cell fitness for cellular therapy by ex vivo activation and ibrutinib
23. Structural basis of selective cannabinoid CB2 receptor activation
24. A novel antifolate suppresses growth of FPGS-deficient cells and overcomes methotrexate resistance
25. Regulation of Adipose Tissue Metabolism by the Endocannabinoid System
26. Piperidine and octahydropyrano[3,4-c] pyridine scaffolds for drug-like molecular libraries of the European Lead Factory
27. Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474
28. Goods and bads of endocannabinoid system as a therapeutic target:Lessons learned after 30 years
29. Endocannabinoid turnover in GtoPdb v.2023.1
30. Chemical genetics strategy to profile kinase target engagement reveals role of FES in neutrophil phagocytosis
31. Disruption of tonic endocannabinoid signalling triggers cellular, behavioural and neuroendocrine responses consistent with a stress response.
32. Inhibition of diacylglycerol lipase β modulates lipid and endocannabinoid levels in the ex vivo human placenta
33. Understanding and Targeting the Endocannabinoid System with Activity‐Based Protein Profiling
34. EFMC – Trends that Link Medicinal Chemistry and Chemical Biology to Translational Drug Discovery
35. Anandamide and other N-acylethanolamines: A class of signaling lipids with therapeutic opportunities
36. Inhibitors of diacylglycerol lipases in neurodegenerative and metabolic disorders
37. Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition
38. EFMC - trends that link medicinal chemistry and chemical biology to translational drug discovery
39. Goods and bads of endocannabinoid system as a therapeutic target: Lessons learned after 30 years
40. Opportunities for Lipid-Based Probes in the Field of Immunology
41. Anti-neuroinflammatory effects of GPR55 antagonists in LPS-activated primary microglial cells
42. Cyclopentitol as a scaffold for a natural product-like compound library for drug discovery
43. Chemical Proteomics Reveals Antibiotic Targets of Oxadiazolones in MRSA
44. 2-AG-Mediated Control of GABAergic Signaling Is Impaired in a Model of Epilepsy
45. Chemical Probes to Control and Visualize Lipid Metabolism in the Brain
46. Comparative Photoaffinity Profiling of Omega-3 Signaling Lipid Probes Reveals Prostaglandin Reductase 1 as a Metabolic Hub in Human Macrophages
47. Disruption of Tonic Endocannabinoid Signaling Triggers the Generation of a Stress Response
48. Live‐Cell Imaging of Sterculic Acid—a Naturally Occurring 1,2‐Cyclopropene Fatty Acid—by Bioorthogonal Reaction with Turn‐On Tetrazine‐Fluorophore Conjugates**
49. Evaluation of different drug classes on transient sciatic nerve injury–depressed marble burying in mice
50. Chemical tools to modulate 2‐arachidonoylglycerol biosynthesis
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