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Your search keyword '"Balzarini Jan"' showing total 9 results
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9 results on '"Balzarini Jan"'

1. Supplementary Figure Legends 1-3 from The Thymidine Phosphorylase Inhibitor 5′-O-Tritylinosine (KIN59) Is an Antiangiogenic Multitarget Fibroblast Growth Factor-2 Antagonist

Author

Liekens, Sandra, primary, Bronckaers, Annelies, primary, Belleri, Mirella, primary, Bugatti, Antonella, primary, Sienaert, Rebecca, primary, Ribatti, Domenico, primary, Nico, Beatrice, primary, Gigante, Alba, primary, Casanova, Elena, primary, Opdenakker, Ghislain, primary, Pérez-Pérez, María-Jesús, primary, Balzarini, Jan, primary, and Presta, Marco, primary

Published
2023
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2. Supplementary Figure 1 from The Thymidine Phosphorylase Inhibitor 5′-O-Tritylinosine (KIN59) Is an Antiangiogenic Multitarget Fibroblast Growth Factor-2 Antagonist

Author

Liekens, Sandra, primary, Bronckaers, Annelies, primary, Belleri, Mirella, primary, Bugatti, Antonella, primary, Sienaert, Rebecca, primary, Ribatti, Domenico, primary, Nico, Beatrice, primary, Gigante, Alba, primary, Casanova, Elena, primary, Opdenakker, Ghislain, primary, Pérez-Pérez, María-Jesús, primary, Balzarini, Jan, primary, and Presta, Marco, primary

Published
2023
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3. Supplementary Figure 3 from The Thymidine Phosphorylase Inhibitor 5′-O-Tritylinosine (KIN59) Is an Antiangiogenic Multitarget Fibroblast Growth Factor-2 Antagonist

Author

Liekens, Sandra, primary, Bronckaers, Annelies, primary, Belleri, Mirella, primary, Bugatti, Antonella, primary, Sienaert, Rebecca, primary, Ribatti, Domenico, primary, Nico, Beatrice, primary, Gigante, Alba, primary, Casanova, Elena, primary, Opdenakker, Ghislain, primary, Pérez-Pérez, María-Jesús, primary, Balzarini, Jan, primary, and Presta, Marco, primary

Published
2023
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4. Data from The Thymidine Phosphorylase Inhibitor 5′-O-Tritylinosine (KIN59) Is an Antiangiogenic Multitarget Fibroblast Growth Factor-2 Antagonist

Author

Liekens, Sandra, primary, Bronckaers, Annelies, primary, Belleri, Mirella, primary, Bugatti, Antonella, primary, Sienaert, Rebecca, primary, Ribatti, Domenico, primary, Nico, Beatrice, primary, Gigante, Alba, primary, Casanova, Elena, primary, Opdenakker, Ghislain, primary, Pérez-Pérez, María-Jesús, primary, Balzarini, Jan, primary, and Presta, Marco, primary

Published
2023
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5. Supplementary Figure 2 from The Thymidine Phosphorylase Inhibitor 5′-O-Tritylinosine (KIN59) Is an Antiangiogenic Multitarget Fibroblast Growth Factor-2 Antagonist

Author

Liekens, Sandra, primary, Bronckaers, Annelies, primary, Belleri, Mirella, primary, Bugatti, Antonella, primary, Sienaert, Rebecca, primary, Ribatti, Domenico, primary, Nico, Beatrice, primary, Gigante, Alba, primary, Casanova, Elena, primary, Opdenakker, Ghislain, primary, Pérez-Pérez, María-Jesús, primary, Balzarini, Jan, primary, and Presta, Marco, primary

Published
2023
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8. Benzothiazole Derivatives as Multifunctional Antioxidant Agents for Skin Damage: Structure–Activity Relationship of a Scaffold Bearing a Five-Membered Ring System

Author

Djuidje, Ernestine Nicaise, primary, Barbari, Riccardo, additional, Baldisserotto, Anna, additional, Durini, Elisa, additional, Sciabica, Sabrina, additional, Balzarini, Jan, additional, Liekens, Sandra, additional, Vertuani, Silvia, additional, and Manfredini, Stefano, additional

Published
2022
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9. 3,5-Bis(benzylidene)-1-[3-(2-hydroxyethylthio)propanoyl]piperidin-4-ones: A Novel Cluster of Potent Tumor-Selective Cytotoxins

Author

Das, Umashankar, Pati, Hari N., Sakagami, Hiroshi, Hashimoto, Ken, Kawase, Masami, Balzarini, Jan, De Clercq, Erik, and Dimmock, Jonathan R.

Abstract

Novel 3,5-bis(benzylidene)-1-[3-(2-hydroxyethylthio)propanoyl]piperidin-4-ones (3a-e)display potent cytotoxicity and a preferential lethality toward various neoplasms compared to some normal cells. The corresponding sulfonic acid analogues 5a−eand an isostere 4demonstrated substantially lower activity. The leads 3dand 3epossess very high activity against colon cancer and leukemia cell lines, caused DNA fragmentation, and activated caspase-3 in HL-60 cells. The enones 3b−ewere well tolerated in a short-term toxicity screen in mice.

Published
2024
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