108 results on '"Spring, David R."'
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2. Unlocking Amides: A General Method for the Self‐Immolative Release of Amide‐Containing Molecules
3. Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late‐Stage Functionalisation
4. Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance
5. Front Cover: Hybrid Androgen Receptor Inhibitors Outperform Enzalutamide and EPI‐001 in in vitro Models of Prostate Cancer Drug Resistance (ChemMedChem 2/2023)
6. Expeditious Total Synthesis of Hemiasterlin through a Convergent Multicomponent Strategy and Its Use in Targeted Cancer Therapeutics
7. Divergent Synthesis of Novel Cylindrocyclophanes that Inhibit Methicillin‐Resistant Staphylococcus aureus (MRSA)
8. Synthesis of Structurally Diverse N-Substituted Quaternary-Carbon-Containing Small Molecules from α,α-Disubstituted Propargyl Amino Esters
9. Cycloaddition Strategies for the Synthesis of Diverse Heterocyclic Spirocycles for Fragment‐Based Drug Discovery
10. Synthesis of Structurally Diverse N-Substituted Quaternary-Carbon-Containing Small Molecules from α,α-Disubstituted Propargyl Amino Esters
11. Two-Component Stapling of Biologically Active and Conformationally Constrained Peptides: Past, Present, and Future
12. Development of a Multifunctional Benzophenone Linker for Peptide Stapling and Photoaffinity Labelling
13. Targeting the Genome-Stability Hub Ctf4 by Stapled-Peptide Design
14. Development of Cell-Permeable, Non-Helical Constrained Peptides to Target a Key Protein-Protein Interaction in Ovarian Cancer
15. Divergent Synthesis of Quinolone Natural Products fromPseudonocardiasp. CL38489
16. ChemInform Abstract: The Reductive Cleavage of Picolinic Amides.
17. Partially Saturated Bicyclic Heteroaromatics as an sp3 -Enriched Fragment Collection
18. A Multidimensional Diversity-Oriented Synthesis Strategy for Structurally Diverse and Complex Macrocycles
19. Multiple-parameter Optimization in Drug Discovery: Example of the 5-HT1B GPCR
20. ChemInform Abstract: Diversity-Oriented Synthesis of Macrocycle Libraries for Drug Discovery and Chemical Biology
21. Development of a Multifunctional Benzophenone Linker for Peptide Stapling and Photoaffinity Labelling
22. The Synthesis of Quinolone Natural Products fromPseudonocardiasp.
23. Double Strain‐Promoted Macrocyclization for the Rapid Selection of Cell‐Active Stapled Peptides
24. ChemInform Abstract: Enantioselective Synthesis of Chromanones via a Peptidic Phosphane Catalyzed Rauhut-Currier Reaction.
25. ChemInform Abstract: Synthesis of a Novel Polycyclic Ring Scaffold with Antimitotic Properties via a Selective Domino Heck-Suzuki Reaction.
26. ChemInform Abstract: Diversity-Oriented Synthesis of Drug-Like Macrocyclic Scaffolds Using an Orthogonal Organo- and Metal Catalysis Strategy.
27. ChemInform Abstract: Peptide Stapling Techniques Based on Different Macrocyclization Chemistries
28. ChemInform Abstract: Concise Synthesis of Substituted Quinolizin‐4‐ones by Ring‐Closing Metathesis.
29. ChemInform Abstract: Arene C—H Functionalization Using a Removable/Modifiable or a Traceless Directing Group Strategy
30. Linear Aliphatic Dialkynes as Alternative Linkers for Double-Click Stapling of p53-Derived Peptides
31. Diversity-Oriented Synthesis of Drug-Like Macrocyclic Scaffolds Using an Orthogonal Organo- and Metal Catalysis Strategy
32. Concise Synthesis of Substituted Quinolizin‐4‐ones by Ring‐Closing Metathesis
33. ChemInform Abstract: Concise Copper‐Catalyzed Synthesis of Tricyclic Biaryl Ether‐Linked Aza‐Heterocyclic Ring Systems.
34. ChemInform Abstract: Combating Multidrug-Resistant Bacteria: Current Strategies for the Discovery of Novel Antibacterials
35. Virulence inPectobacterium atrosepticumis regulated by a coincidence circuit involving quorum sensing and the stress alarmone, (p)ppGpp
36. Combating Multidrug‐Resistant Bacteria: Current Strategies for the Discovery of Novel Antibacterials
37. Die Bekämpfung multiresistenter Bakterien: aktuelle Strategien zur Entdeckung neuer Antibiotika
38. ChemInform Abstract: Mild and Efficient Synthesis of Benzo‐Fused Seven‐ and Eight‐Membered Ring Lactams: A Convenient Approach to Biologically Interesting Chemotypes.
39. ChemInform Abstract: Palladium‐Catalyzed Cross‐Coupling of Vinyldisiloxanes with Benzylic and Allylic Halides and Sulfonates.
40. Using Ligand-Mapping Simulations to Design a Ligand Selectively Targeting a Cryptic Surface Pocket of Polo-Like Kinase 1
41. ChemInform Abstract: Diversity‐Oriented Synthesis: Producing Chemical Tools for Dissecting Biology
42. Palladium‐Catalysed Cross‐Coupling of Vinyldisiloxanes with Benzylic and Allylic Halides and Sulfonates
43. ChemInform Abstract: Diversity‐Oriented Synthesis
44. ChemInform Abstract: Palladium-Catalyzed Cross-Coupling of Organosilicon Reagents
45. ChemInform Abstract: Synthesis of Highly Substituted Symmetrical 1,3‐Dienes via Organocuprate Oxidation.
46. ChemInform Abstract: Aryl—Aryl Bond Formation by the Fluoride‐Free Cross‐Coupling of Aryldisiloxanes with Aryl Bromides.
47. A Concise Total Synthesis of Deoxyschizandrin and Exploration of Its Antiproliferative Effects and those of Structurally Related Derivatives
48. ChemInform Abstract: Chemical Genetics
49. Aryl-Aryl Bond Formation by the Fluoride-Free Cross-Coupling of Aryldisiloxanes with Aryl Bromides
50. ChemInform Abstract: Novel and Efficient Copper‐Catalyzed Synthesis of Nitrogen‐Linked Medium‐Ring Biaryls.
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