510 results on '"van der Stelt, Mario"'
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102. Metabolic Fate of Endocannabinoids
103. The endocannabinoid system in the basal ganglia and in the mesolimbic reward system: implications for neurological and psychiatric disorders
104. In Vivo Excitotoxicity Induced by Ouabain, a Na+/K+-ATPase Inhibitor
105. Endocannabinoid turnover (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database
106. Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors
107. Comprehensive structure-activity-relationship of azaindoles as highly potent FLT3 inhibitors
108. High Fat Diet Increases Circulating Endocannabinoids Accompanied by Increased Synthesis Enzymes in Adipose Tissue
109. Activity-Based Protein Profiling Identifies α-Ketoamides as Inhibitors for Phospholipase A2 Group XVI
110. Gene Expression o Endocannabinoid System Components in Skeletal Muscle and Adipose Tissue of South Asians and White Caucasians with Overweight
111. Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N‑Acylphosphatidylethanolamine Phospholipase D.
112. A Fluorescence Polarization Activity-Based Protein Profiling Assay in the Discovery of Potent, Selective Inhibitors for Human Nonlysosomal Glucosylceramidase
113. Cannabinoid CB receptor ligand profiling reveals biased signalling and off-target activity
114. Endocannabinoid contributions to alcohol habits and motivation: Relevance to treatment.
115. Drug Discovery Maps, a Machine Learning Model That Visualizes and Predicts Kinome–Inhibitor Interaction Landscapes
116. Activity-Based Protein Profiling Delivers Selective Drug Candidate ABX-1431, a Monoacylglycerol Lipase Inhibitor, To Control Lipid Metabolism in Neurological Disorders
117. Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors
118. An Affinity-Based Probe for the Human Adenosine A2A Receptor
119. Gene Expression of Endocannabinoid System Components in Skeletal Muscle and Adipose Tissue of South Asians and White Caucasians with Overweight
120. Chemical Proteomic Analysis of Serine Hydrolase Activity in Niemann-Pick Type C Mouse Brain
121. 2-Arachidonoylglycerol: A signaling lipid with manifold actions in the brain
122. Development of a Cannabinoid-Based Photoaffinity Probe to Determine the Δ8/9-Tetrahydrocannabinol Protein Interaction Landscape in Neuroblastoma Cells
123. Structure-kinetic relationship studies of cannabinoid CB 2 receptor agonists reveal substituent-specific lipophilic effects on residence time
124. Mapping in vivo target interaction profiles of covalent inhibitors using chemical proteomics with label-free quantification
125. Localization of the cannabinoid type-1 receptor in subcellular astrocyte compartments of mutant mouse hippocampus
126. Selective Photoaffinity Probe That Enables Assessment of Cannabinoid CB2 Receptor Expression and Ligand Engagement in Human Cells
127. Activity-Based Protein Profiling
128. Two-step activity-based protein profiling of diacylglycerol lipase
129. A Fluorescence Polarization Activity-Based Protein Profiling Assay in the Discovery of Potent, Selective Inhibitors for Human Nonlysosomal Glucosylceramidase
130. Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474
131. The Chemical Biology‐Medicinal Chemistry Continuum: EFMC′s Vision.
132. Asymmetric Synthesis of Lysine Analogues with Reduced Basicity, and their Incorporation into Proteasome Inhibitors
133. Endocannabinoid tone is higher in healthy lean South Asian than white Caucasian men
134. Chemical tools to modulate 2-arachidonoylglycerol biosynthesis
135. A Novel Selective Inverse Agonist of the CB2 Receptor as a Radiolabeled Tool Compound for Kinetic Binding Studies
136. Quantitative profiling of endocannabinoids and related N-acylethanolamines in human CSF using nano LC-MS/MS
137. Chemical Proteomics Maps Brain Region Specific Activity of Endocannabinoid Hydrolases
138. Novel activity-based probes for N-acylethanolamine acid amidase
139. Chiral disubstituted piperidinyl ureas: a class of dual diacylglycerol lipase-α and ABHD6 inhibitors
140. Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding
141. Drug Discovery Maps, a Machine Learning Model That Visualizes and Predicts Kinome–Inhibitor Interaction Landscapes.
142. Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors
143. Targeting IGF1R/Insr Pathway with Approved ALK-Inhibitors Overcomes Proteasome Inhibitor Resistance in Multiple Myeloma
144. Structure-Based Design of β5c Selective Inhibitors of Human Constitutive Proteasomes
145. Photo-crosslinking of clinically relevant kinases using H89-derived photo-affinity probes
146. Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition
147. Identification of an allosteric binding site for RORγt inhibition
148. Comprehensive Analysis of Structure–Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α Inhibitors
149. An Affinity-Based Probe for the Human Adenosine A2A Receptor.
150. Development of a Cannabinoid-Based Photoaffinity Probe to Determine the Δ8/9-Tetrahydrocannabinol Protein Interaction Landscape in Neuroblastoma Cells.
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