144 results on '"Bair, Kenneth W."'
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2. Molecular basis of USP7 inhibition by selective small-molecule inhibitors
3. 2-((Arylmethyl)Amino)-1, 3-Propanediols (AMAPS); Discovery, Selection and Development of Four Clinical Candidates
4. Hairpin versus extended DNA binding of a substituted beta-alanine linked polyamide
5. Total syntheses of bengamides B and E
6. Bengamides revisited: new structures and antitumor studies
7. Discovery and optimization of novel piperazines as potent inhibitors of fatty acid synthase (FASN)
8. Small molecule blockade of transcriptional coactivation of the hypoxia-inducible factor pathway
9. An efficient multiple-exposure analysis of the toxicity of crisnatol, a DNA intercalator in phase II clinical trials
10. Effects of isomeric 2-(Arylmethylamino)-1,3-propanediols (AMAPs) and clinically established agents on macromolecular synthesis in P388 and MCF-7 cells
11. Proteomics-based Target Identification: BENGAMIDES AS A NEW CLASS OF METHIONINE AMINOPEPTIDASE INHIBITORS
12. Discovery and Optimization of Quinolinone Derivatives as Potent, Selective, and Orally Bioavailable Mutant Isocitrate Dehydrogenase 1 (mIDH1) Inhibitors
13. Total synthesis of (plus or minus)-illudin M
14. Psammaplins from the sponge Pseudoceratina purpurea: inhibition of both histone deacetylase and DNA methyltransferase
15. Discovery of potent and efficacious cyanoguanidine-containing nicotinamide phosphoribosyltransferase (Nampt) inhibitors
16. Identification of amides derived from 1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
17. Identification of 2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-derived ureas as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
18. Discovery of potent and efficacious urea-containing nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with reduced CYP2C9 inhibition properties
19. Minimizing CYP2C9 Inhibition of Exposed-Pyridine NAMPT (Nicotinamide Phosphoribosyltransferase) Inhibitors
20. Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility
21. Structural Basis for Resistance to Diverse Classes of NAMPT Inhibitors
22. Fragment-Based Identification of Amides Derived from trans-2-(Pyridin-3-yl)cyclopropanecarboxylic Acid as Potent Inhibitors of Human Nicotinamide Phosphoribosyltransferase (NAMPT)
23. Structure-Based Discovery of Novel Amide-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
24. Structure-Based Identification of Ureas as Novel Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
25. ChemInform Abstract: Bengamides Revisited: New Structures and Antitumor Studies.
26. N-Hydroxy-3-phenyl-2-propenamides as Novel Inhibitors of Human Histone Deacetylase with in Vivo Antitumor Activity: Discovery of (2E)-N-Hydroxy-3-[4-[[(2-hydroxyethyl)[2-(1H-indol-3-yl)ethyl]amino]methyl]phenyl]-2-propenamide (NVP-LAQ824)
27. Synthesis and DNA Binding Properties of Saturated Distamycin Analogues.
28. Synthesis and DNA binding properties of saturated distamycin analogues
29. Hairpin versus Extended DNA Binding of a Substituted β-Alanine Linked Polyamide
30. Inhibitors of Human Histone Deacetylase: Synthesis and Enzyme and Cellular Activity of Straight Chain Hydroxamates
31. Synthesis and Antitumor Activity of Ester-Modified Analogues of Bengamide B
32. Identification of E2F-1/Cyclin A antagonists
33. Fragment-Based Identificationof Amides Derived from trans-2-(Pyridin-3-yl)cyclopropanecarboxylicAcid as PotentInhibitors of Human Nicotinamide Phosphoribosyltransferase (NAMPT).
34. Selective Killing of Cancer Cells based on Derepression of E2F
35. Structural and Conformational Requirements for High-Affinity Binding to the SH2 Domain of Grb2
36. Synthesis of Isodehydroilludin M
37. Solid Phase Synthesis of β-Peptides via Arndt-Eistert Homologation of Fmoc-Protected Amino Acid Diazoketones
38. Synthesis of Tricyclic Analogues of Illudin M
39. Synthesis of Bicyclic Analogues of Dehydroilludin M
40. Design, synthesis, and antitumor activity of bicyclic and isomeric analogues of illudin M
41. Total Synthesis of (.+-.)-Illudin M
42. Retrospective Review: Cancer Drug Development: Current Research and Patents - 1992 - Part 1
43. Patent Update: Cancer Drug Development: Current Research and Patents - 1991 - Part 2
44. Patent Update: Cancer Drug Development: Current Research and Patents in 1991 - Part 1
45. Polyploidy induction as a consequence of topoisomerase inhibition
46. Phase I evaluation of 773U82 HCI, a member of a new class of DNA intercalators
47. 2-[(Arylmethyl)amino]-2-methyl-1,3-propanediol DNA intercalators. An examination of the effects of aromatic ring variation on antitumor activity and DNA binding
48. [(1-Pyrenylmethyl)amino] alcohols, a new class of antitumor DNA intercalators. Discovery and initial amine side chain structure-activity studies
49. USES OF THE TRIFYL GROUP IN ORGANIC SYNTHESIS. A REVIEW.
50. Solid Phase Synthesis of β-Peptides viaArndt-Eistert Homologation of Fmoc-Protected Amino Acid Diazoketones
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