701 results on '"Besson, Thierry"'
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2. Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia
3. Contribution of Professor Charles W. Rees to the development of the chemistry of disulfur dichloride
4. Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinases
5. Relieving DYRK1A repression of MKL1 confers an adult-like phenotype to human infantile megakaryocytes
6. Synthesis of Thiazole-fused Tricyclic Quinazolinone Alkaloids and Their Derivatives.
7. Synthesis of Trifunctional Thiazole-Fused Anthranilonitrile and Anthranilic Acid Derivatives
8. Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinasesElectronic supplementary information (ESI) available: 1H and 13C NMR spectra, HRMS spectra 1b–p, amino-acid sequence alignment of eqBuChE and hBuChE. See DOI: https://doi.org/10.1039/d3md00708a
9. Photocatalyst-Free, Visible-Light-Mediated C–H Perfluoroalkylation of Quinazolin-4(3 H)-ones with perfluoroalkyl Iodides.
10. Synthesis of Trifunctional Thiazole-Fused Anthranilonitrile and Anthranilic Acid Derivatives.
11. Photocatalyst-Free, Visible-Light-Mediated C–H Perfluoroalkylation of Quinazolin-4(3H)-ones with perfluoroalkyl Iodides
12. DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3
13. Synthesis and molecular modelling studies of 8-arylpyrido[3′,2′:4,5]thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors
14. Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core
15. Synthesis of 2-Cyanobenzothiazoles via Pd-Catalyzed/Cu-Assisted C-H Functionalization/Intramolecular C-S Bond Formation from N-Arylcyanothioformamides
16. Pharmacologic Inhibition of DYRK1A Results in Hyperactivation and Hyperphosphorylation of MYC and ERK Rendering KMT2A-R ALL Cells Sensitive to BCL2 Inhibition
17. Pharmacologic Inhibition of DYRK1A Results in MYC Hyperactivation and ERK Hyperphosphorylation rendering KMT2A-R ALL Cells Sensitive to BCL2 Inhibition
18. Monitoring of Catalyst-Free Microwave-Assisted MCR-Type Synthesis of 2-Amino-3-cyano-4H-chromene Derivatives Using Raman Spectrometry
19. Microwave-assisted synthesis of novel N-(4-phenylthiazol-2-yl)-benzo[d]thiazole-, thiazolo[4,5-b]pyridine-, thiazolo[5,4-b]pyridine- and benzo[d]oxazole-2-carboximidamides inspired by marine topsentines and nortopsentines
20. Rational multistep synthesis of a novel polyfunctionalized benzo[d]thiazole and its thiazolo[5,4-b]pyridine analogue
21. Microwave-Assisted Synthesis of Sulfur and Nitrogen-Containing Heterocycles
22. Therapeutic antibody glycosylation impacts antigen recognition and immunogenicity
23. Radiosynthesis of [11C]EHT1610, a potential radioligand for quantification of cerebral DYRK1A by PET imaging
24. Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs
25. Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases
26. Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors
27. Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core.
28. Synthesis of novel 7-oxo and 7-hydroxy trifluoroallocolchicinoids with cytotoxic effect
29. Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-d], [3,2-d], [3,4-d] and [4,3-d]pyrimidine Derivatives
30. Structure of Pb2+/dCMP and Pb2+/CMP complexes as characterized by tandem mass spectrometry and IRMPD spectroscopy
31. Microwave-assisted thermal decomposition of formamide: a tool for coupling a pyrimidine ring with an aromatic partner
32. Pharmacologic Inhibition of DYRK1A Results in Hyperactivation and Hyperphosphorylation of MYC and ERK Rendering KMT2A-R ALL Cells Sensitive to BCL2 Inhibition
33. Microwave-assisted copper catalyzed C-H arylation of bioactive pyrimidinones using diaryliodoniums salts
34. Monitoring of Catalyst-Free Microwave-Assisted MCR-Type Synthesis of 2-Amino-3-cyano-4 H -chromene Derivatives Using Raman Spectrometry.
35. Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts
36. Référentiel des compétences de chimie thérapeutique pertinentes pour l’exercice contemporain de la pharmacie
37. A novel DYRK1A (Dual specificity tyrosine phosphorylation-regulated kinase 1A) inhibitor for the treatment of Alzheimerʼs disease: effect on Tau and amyloid pathologies in vitro
38. Synthesis and antitumoral activity of novel thiazolobenzotriazole, thiazoloindolo[3,2- c]quinoline and quinolinoquinoline derivatives
39. Synthesis and kinase inhibitory activity of novel substituted indigoids
40. Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-a][1,3,5]triazines
41. Novel 9-oxo-thiazolo[5,4- f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies
42. Demonstration of Green Solvent Performance on O,S,N-Heterocycles Synthesis: Metal-Free Click Chemistry and Buchwald—Hartwig Coupling
43. On the origin of some cubebene derivatives--Diels-Alder adducts and the diene structures of solidago compounds
44. Synthesis and antiproliferative activity of clausine E, mukonine, and koenoline bioisosteres
45. Synthesis of latonduine derivatives via intramolecular Heck reaction
46. Synthesis of novel 2,3-substituted quinazolin-4-ones by condensation of alkyl or aromatic diamines with 5-( N-arylimino)-4-chloro-5 H-1,2,3-dithiazoles
47. Copper-Catalyzed C–H Arylation of Fused-Pyrimidinone Derivatives Using Diaryliodonium Salts
48. Exploring kinase inhibition properties of 9<em>H</em>-pyrimido[5,4-<em>b</em>]- and [4,5-<em>b</em>]indol-4-amine derivatives
49. Synthesis of potential bioactive benzo-, pyrido-, or pyrazinothieno[3,2-d]pyrimidin- 4-amine analogs of MPC-6827
50. DYRK1A Is Required to Alleviate Replication Stress in KMT2A-Rearranged Acute Lymphoblastic Leukemia
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