33 results on '"Blaquiere, Nicole"'
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2. Filling a nick in NIK: extending the half-life of a NIK inhibitor through structure-based drug design
3. Filling a Nick in NIK: Extending the Half-Life of a NIK Inhibitor Through Structure-Based Drug Design
4. Discovery and Preclinical Pharmacology of INE963, a Potent and Fast-Acting Blood-Stage Antimalarial with a High Barrier to Resistance and Potential for Single-Dose Cures in Uncomplicated Malaria
5. Primary Amine Tethered Small Molecules Promote the Degradation of X-Linked Inhibitor of Apoptosis Protein
6. Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα)
7. Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1: Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties
8. Monomeric Targeted Protein Degraders
9. Medicinal Chemistry of Inhibiting RING-Type E3 Ubiquitin Ligases
10. Scaffold-Hopping Approach To Discover Potent, Selective, and Efficacious Inhibitors of NF-κB Inducing Kinase
11. NF-κB inducing kinase is a therapeutic target for systemic lupus erythematosus
12. Decarboxylative ketone aldol reactions: development and mechanistic evaluation under metal-free conditions
13. Ruthenium-catalyzed dehydrogenation of ammonia boranes
14. Selective inhibition of NF-kB inducing kinase (NIK) is therapeutically efficacious in IFNα-accelerated lupus nephritis prone mice
15. Structure-Based Design of Tricyclic NF-κB Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K)
16. Discovery of thiazolobenzoxepin PI3-kinase inhibitors that spare the PI3-kinase β isoform
17. Cis-Amide isosteric replacement in thienobenzoxepin inhibitors of PI3-kinase
18. Part I The development and mechanistic study of a biomimetic decarboxylative aldol reaction Part II Ruthenium-catalyzed dehydrogenation of ammonia-boranes
19. Development of a tripartite solvent blend for sustainable chromatography
20. Discovery of 2-{3-[2-(1-Isopropyl-3-methyl-1H-1,2–4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl]-1H-pyrazol-1-yl}-2-methylpropanamide (GDC-0032): A β-Sparing Phosphoinositide 3-Kinase Inhibitor with High Unbound Exposure and Robust in Vivo Antitumor Activity
21. Abstract DDT02-01: Discovery of GDC-0032: A beta-sparing PI3K inhibitor active against PIK3CA mutant tumors.
22. ChemInform Abstract: Heteroarylation of Azine N-Oxides.
23. Heteroarylation of Azine N-Oxides
24. ChemInform Abstract: Rapid Synthesis of 1,3,5‐Substituted 1,2,4‐Triazoles from Carboxylic Acids, Amidines, and Hydrazines.
25. Rapid Synthesis of 1,3,5-Substituted 1,2,4-Triazoles from Carboxylic Acids, Amidines, and Hydrazines
26. ChemInform Abstract: Four‐Component Synthesis of Fully Substituted 1,2,4‐Triazoles.
27. Four‐Component Synthesis of Fully Substituted 1,2,4‐Triazoles
28. Four‐Component Synthesis of Fully Substituted 1,2,4‐Triazoles
29. Aporphine Alkaloid Synthesis and Diversification via Direct Arylation.
30. Direct Intramolecular Arylation of Unactivated Arenes: Application to the Synthesis of Aporphine Alkaloids.
31. Discoveryof 2-{3-[2-(1-Isopropyl-3-methyl-1H-1,2–4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl]-1H-pyrazol-1-yl}-2-methylpropanamide(GDC-0032): A β-Sparing Phosphoinositide 3-KinaseInhibitor with High Unbound...
32. Aporphine Alkaloid Synthesis and Diversification via Direct Arylation
33. Four-component synthesis of fully substituted 1,2,4-triazoles.
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