2,143 results on '"Hruby, Victor J."'
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2. Melanocortin 3 receptor activation with [D-Trp8]-γ-MSH suppresses inflammation in apolipoprotein E deficient mice
3. Replacement of Arg with Nle and modified D-Phe in the core sequence of MSHs, Ac-His-D-Phe-Arg-Trp-NH2, leads to hMC1R selectivity and pigmentation
4. Ψ and χ Angle Constrains at the C-Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH2 Lead to Potent and Selective Agonists at hMC1R and hMC4R
5. The Melanocortin-1 Receptor Gene Mediates Female-Specific Mechanisms of Analgesia in Mice and Humans
6. Melanocortin receptors in GtoPdb v.2023.1
7. Supplementary Figures 1-6 from Enhanced targeting with heterobivalent ligands
8. Supplementary Table S1 from Gene expression profiling-based identification of cell-surface targets for developing multimeric ligands in pancreatic cancer
9. Data from Gene expression profiling-based identification of cell-surface targets for developing multimeric ligands in pancreatic cancer
10. Melanotropic Peptide-Conjugated Beads for Microscopic Visualization and Characterization of Melanoma Melanotropin Receptors
11. Design synthesis and structure–activity relationship of 5-substituted (tetrahydronaphthalen-2yl)methyl with N-phenyl-N-(piperidin-2-yl)propionamide derivatives as opioid ligands
12. Melanotropin Receptors and Signal Transduction
13. Cyclic, Conformationally Constrained Melanotropin Analogs: Structure-Function and Conformational Relationships
14. Melanotropin Three-Dimensional Structural Studies by Physical Methods and Computer-Assisted Molecular Modeling
15. Adjuvants in Cancer Vaccines - Progress and Challenges
16. Discovery of 5-substituted tetrahydronaphthalen-2yl-methyl with N-phenyl-N-(piperidin-4-yl)propionamide derivatives as potent opioid receptor ligands
17. Design, synthesis, and biological evaluation of a series of bifunctional ligands of opioids/SSRIs
18. Simple size-selective separation and microscopic characterization of Phe–Phe nanotubes and study of its internalization inside CHO cells
19. Synthesis and evaluation of bivalent ligands for binding to the human melanocortin-4 receptor
20. Delta Opioid Receptor Function
21. Protection against β‐amyloid neurotoxicity by a non‐toxic endogenous N‐terminal β‐amyloid fragment and its active hexapeptide core sequence
22. New Paradigms and Tools in Drug Design for Pain and Addiction
23. Ψ and χ Angle Constrains at the C‑Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His‑d‑Phe-Arg-Trp-NH2 Lead to Potent and Selective Agonists at hMC1R and hMC4R.
24. Examination of the Role of Lipid Rafts in GPCR Signal Transduction Using Plasmon Waveguide Resonance (PWR) Spectroscopy
25. Novel fentanyl-based dual μ/δ-opioid agonists for the treatment of acute and chronic pain
26. MC4R biased signalling and the conformational basis of biological function selections
27. Synthesis and Characterization of Time-resolved Fluorescence Probes for Evaluation of Competitive Binding to Melanocortin Receptors
28. Perspectives for the new peptide millennium
29. Design of a δ opioid peptide mimetic based on a topographically constrained cyclic enkephalin
30. Heterobivalent ligands target cell-surface receptor combinations in vivo
31. The Molecular Pharmacology of Alpha-Melanocyte Stimulating Hormone : Structure—Activity Relationships for Melanotropins at Melanocortin Receptors
32. New Perspective in Peptide Chemistry by N-Alkylation
33. CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists
34. Entrap and release of Phe–Phe nanotubes in sol–gel derived silicate matrix: study through nanosilver interaction
35. The Potential Application of Melanotropin Ligands for the Treatment of Obesity and Related Disorders: Potential and Problems
36. Discovery and Development of Novel Melanogenic Drugs : Melanotan-I and -II
37. Design, Synthesis, and Evaluation of Piperazine-Based Small Molecule Peptide Mimetics Targeting the Melanocortin Receptors
38. Understanding BBB Transport using Glycosylated Enkephalins and Endorphins
39. Ψ and χ Angle Constrains at the C-Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH2Lead to Potent and Selective Agonists at hMC1R and hMC4R
40. Conformational study on cyclic melanocortin ligands and new insight into their binding mode at the MC4 receptor
41. Synthesis and biological evaluation of new opioid agonist and neurokinin-1 antagonist bivalent ligands
42. The Design and Synthesis of Long-Acting Oxytocin Antagonists Substituted in Positions 2, 7, and 8
43. Practical glycopeptide analgesics: Blood-brain barrier transport and binding of glycosylated enkephalin analogs
44. Efficacy: What is it, and why you should care
45. Stereoselective synthesis of highly topographically constrained β-isopropyl substituted aromatic amino acids
46. Design of novel melanotropin antagonists and agonists for the recently discovered MC3, MC4 and MC5 receptors and their use to determine new biological roles
47. α-Helical Glycopeptide Analgesics: β-Endorphin Mimics with Good in vivo Potency
48. Rational Approach to the Design of Bioactive Peptidomimetics: Recent Developments in Opioid Agonist Peptides
49. Optimization of time-resolved fluorescence assay for detection of europium–tetraazacyclododecyltetraacetic acid-labeled ligand–receptor interactions
50. Use of plasmon waveguide resonance (PWR) spectroscopy for examining binding, signaling and lipid domain partitioning of membrane proteins
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