176 results on '"Jarvest, Richard L."'
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2. 6-Alkylquinolone-3-carboxylic acid tethered to macrolides synthesis and antimicrobial profile
3. Linear and Macrocyclic Hepatitis C Virus Protease Inhibitors: Inhibitor Design and Macrocyclization Strategies for HCV Protease and Related Targets
4. Famciclovir
5. New atropisomeric biaryl derivatives of 4-aminopyridine—identification of an improved nucleophilic catalyst for asymmetric acylation of sec-alcohols
6. Interaction of tyrosyl aryl dipeptides with S. aureus tyrosyl tRNA synthetase: Inhibition and crystal structure of a complex
7. Inhibition of human cytomegalovirus protease by enedione derivatives of thieno[2,3-d]oxazinones through a novel dual acylation/alkylation mechanism
8. Inhibition of herpes proteases and antiviral activity of 2-substituted thieno[2,3-d]oxazinones
9. Concise, synthesis, preparation resolution, absolute configuration determination, and applications of an atropisomeric biaryl catalysts for asymmetric acylation
10. Synthesis and antiviral activity of novel HCV NS3 protease inhibitors with P4 capping groups
11. Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties
12. Chiral [16O, 17O, 18O] Phosphate Monoesters for Determining the Stereochemical Course of Phosphokinases
13. Synthesis and evaluation of novel α-amino cyclic boronates as inhibitors of HCV NS3 protease
14. Novel macrocyclic HCV NS3 protease inhibitors derived from α-amino cyclic boronates
15. Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 protease
16. Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 protease
17. Discovery of Novel Urea-Based Hepatitis C Protease Inhibitors with High Potency against Protease-Inhibitor-Resistant Mutants
18. ChemInform Abstract: Aminoalkyl Adenylate and Aminoacyl Sulfamate Intermediate Analogues Differing Greatly in Affinity for Their Cognate Staphylococcus aureus Aminoacyl tRNA Synthetases
19. ChemInform Abstract: Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Carbocyclic Analogues of the Natural Product SB-219383.
20. Optimization of Novel Acyl Pyrrolidine Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase Leading to a Development Candidate
21. Discovery and optimisation of potent, selective, ethanolamine inhibitors of bacterial phenylalanyl tRNA synthetase
22. Definition of the Heterocyclic Pharmacophore of Bacterial Methionyl tRNA Synthetase Inhibitors: Potent Antibacterially Active Non‐quinolone Analogues
23. New Atropisomeric Biaryl Derivatives of 4‐Aminopyridine—Identification of an Improved Nucleophilic Catalyst for Asymmetric Acylation of sec‐Alcohols.
24. Definition of the heterocyclic pharmacophore of bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues
25. Optimization of Aryl Substitution Leading to Potent Methionyl tRNA Synthetase Inhibitors with Excellent Gram-Positive Antibacterial Activity.
26. Variable Sensitivity to Bacterial Methionyl-tRNA Synthetase Inhibitors Reveals Subpopulations of Streptococcus pneumoniae with Two Distinct Methionyl-tRNA Synthetase Genes
27. Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-Positive antibacterial activity
28. The Antimicrobial Natural Product Chuangxinmycin and Some Synthetic Analogues Are Potent and Selective Inhibitors of Bacterial Tryptophanyl tRNA Synthetase.
29. Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity
30. The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase
31. Nanomolar Inhibitors of Staphylococcus aureus Methionyl tRNA Synthetase with Potent Antibacterial Activity against Gram-Positive Pathogens
32. Crystal structure of Staphylococcus aureus tyrosyl‐tRNA synthetase in complex with a class of potent and specific inhibitors
33. Lewis-acid catalysed arylation of the hydroxyamino sugar moiety of the natural product SB-219383
34. Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Carbocyclic Analogues of the Natural Product SB-219383
35. ChemInform Abstract: Synthetic Analogues of SB‐219383. Novel C‐Glycosyl Peptides as Inhibitors of Tyrosyl tRNA Synthase.
36. ChemInform Abstract: Synthesis and Activity of Analogues of SB-219383: Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase.
37. Synthetic analogues of SB-219383. Novel C-glycosyl peptides as inhibitors of tyrosyl tRNA synthetase
38. Potent synthetic inhibitors of tyrosyl tRNA synthetase derived from C-pyranosyl analogues of SB-219383
39. ChemInform Abstract: Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Four Stereoisomeric Analogues of the Natural Product SB-219383.
40. Inhibitors of bacterial tyrosyl tRNA synthetase: synthesis of four stereoisomeric analogues of the natural product SB-219383
41. Aminoalkyl adenylate and aminoacyl sulfamate intermediate analogues differing greatly in affinity for their cognate Staphylococcus aureus aminoacyl tRNA synthetases
42. ChemInform Abstract: The Synthesis of 5‐Alkoxy and 5‐Amino Substituted Thiophenes.
43. The synthesis of 5-alkoxy and 5-amino substituted thiophenes
44. Synthesis and Activity of Analogues of SB-219383. Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase.
45. ChemInform Abstract: Inhibition of Herpes Proteases and Antiviral Activity of 2‐Substituted Thieno[2,3‐d]oxazinones.
46. Exploring the active site of herpes simplex virus type-1 thymidine kinase by X-ray crystallography of complexes with aciclovir and other ligands
47. Potent selective thienoxazinone inhibitors of herpes proteases
48. Novel, selective mechanism-based inhibitors of the herpes proteases
49. Inhibition of HSV-1 protease by benzoxazinones
50. Structure-directed discovery of an inhibitor of the binding of HIV GP120 to the CD4 receptor
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