288 results on '"Kakuta, Hiroki"'
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2. Simple Fluorescence Labeling Method Enables Detection of Intracellular Distribution and Expression Level of Retinoid X Receptors
3. Direct evaluation of polarity of the ligand binding pocket in retinoid X receptor using a fluorescent solvatochromic agonist
4. Structural basis for the full and partial agonist activities of retinoid X receptor α ligands with an iso-butoxy and an isopropyl group
5. A retinoid X receptor partial agonist attenuates pulmonary emphysema and airway inflammation
6. Supplementary figures #1-#15 from Strategy for Tumor-Selective Disruption of Androgen Receptor Function in the Spectrum of Prostate Cancer
7. Supplementary Tables from Strategy for Tumor-Selective Disruption of Androgen Receptor Function in the Spectrum of Prostate Cancer
8. Ligand Screening System for the RXRα Heterodimer Using the Fluorescence RXR Agonist CU-6PMN
9. Reversal of established liver fibrosis by IC-2-engineered mesenchymal stem cell sheets
10. Analysis of absorption-enhancing mechanisms for combinatorial use of spermine with sodium taurocholate in Caco-2 cells
11. Teratogenicity and Fetal-Transfer Assessment of the Retinoid X Receptor Agonist Bexarotene
12. Development of Scaled-Up Synthetic Method for Retinoid X Receptor Agonist NEt-3IB Contributing to Sustainable Development Goals
13. Relevance of nuclear receptor expression in a Tchreg cell line, HOZOT: RXRα and PPARγ negatively regulate IFN-γ production
14. Identification of a Vitamin-D Receptor Antagonist, MeTC7, which Inhibits the Growth of Xenograft and Transgenic Tumors In Vivo
15. Development of Scaled-Up Synthetic Method for Retinoid X Receptor Agonist NEt-3IB Contributing to Sustainable Development Goals
16. Modified SPEA2 for Probabilistic Reliability Assessment in Smart Grids
17. Replacement of the hydrophobic part of 9- cis-retinoic acid with cyclic terpenoid moiety results in RXR-selective agonistic activity
18. Increased Molecular Flexibility Widens the Gap between Ki and Kd values in Screening for Retinoid X Receptor Modulators
19. A Retinoid X Receptor Agonist Directed to the Large Intestine Ameliorates T-Cell-Mediated Colitis in Mice
20. Fluorescence properties of retinoid X receptor antagonist NEt-SB
21. Creation of Fluorescent RXR Antagonists Based on CBTF-EE and Application to a Fluorescence Polarization Binding Assay
22. A Retinoid X Receptor Agonist Directed to the Large Intestine Ameliorates T-Cell-Mediated Colitis in Mice
23. Design and synthesis of benzenesulfonanilides active against methicillin-resistant Staphylococcus aureus and vancomycin-resistant Enterococcus
24. Pyridinium cationic-dimer antimalarials, unlike chloroquine, act selectively between the schizont stage and the ring stage of Plasmodium falciparum
25. Involvement of glucocorticoid receptor activation on anti-inflammatory effect induced by peroxisome proliferator-activated receptor γ agonist in mice
26. In vitro anti-proliferative and anti-angiogenic activities of thalidomide dithiocarbamate analogs
27. In Vivo Receptor Visualization and Evaluation of Receptor Occupancy with Positron Emission Tomography
28. Analgesic agents without gastric damage: Design and synthesis of structurally simple benzenesulfonanilide-type cyclooxygenase-1-selective inhibitors
29. Convenient Retinoid X Receptor Binding Assay Based on Fluorescence Change of the Antagonist NEt-C343
30. Discovery of a “Gatekeeper” Antagonist that Blocks Entry Pathway to Retinoid X Receptors (RXRs) without Allosteric Ligand Inhibition in Permissive RXR Heterodimers
31. 3H-Imidazo[4,5-b]pyridine-6-carboxylic acid derivatives as rexinoids with reduced teratogenicity
32. An Arylidene-Thiazolidinedione Derivative, GPU-4, without PPARγ Activation, Reduces Retinal Neovascularization
33. Paclitaxel and Sorafenib: The Effective Combination of Suppressing the Self-Renewal of Cancer Stem Cells
34. Ordering Phase Transition with Symmetry-Breaking from Disorder over Non-Equivalent Sites: Calorimetric and Crystallographic Study of Crystalline d-Sorbose
35. Maternal gut microbiota in pregnancy influences offspring metabolic phenotype in mice
36. Effect of 5-aminosalicylate on allergic rhinitis model in mice
37. Additional file 1: of A retinoid X receptor partial agonist attenuates pulmonary emphysema and airway inflammation
38. Syntheses of Thiopyrone and Pyrone Derivatives by Photocyclization Reaction of 3-Aryl-2-([l]benzothien-3-yl)propenoic Acids
39. A partial agonist for retinoid X receptor mitigates experimental colitis
40. Towards Further Sharing of Knowledge and Activities on Standards of Quality Assurance (QA) across Industry, Academia and Government to Promote Research Integrity and Accelerate Drug Discovery
41. Competitive Binding Assay with an Umbelliferone-Based Fluorescent Rexinoid for Retinoid X Receptor Ligand Screening
42. Fluorine-18 (18F)-labeled retinoid x receptor (RXR) partial agonist whose tissue transferability is affected by other RXR ligands
43. Problems with Laboratory Notebooks in Academia and How to Resolve Them
44. Correction to Synthesis of 11C-Labeled RXR Partial Agonist 1-[(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)amino]benzotriazole-5-carboxylic Acid (CBt-PMN) by Direct [11C]Carbon Dioxide Fixation via Organolithiation of Trialkyltin Precursor and PET Imaging Thereof
45. A partial agonist for retinoid X receptor mitigates experimental colitis
46. Dual conformation of the ligand induces the partial agonistic activity of retinoid X receptor α (RXRα)
47. Strategy for Tumor-Selective Disruption of Androgen Receptor Function in the Spectrum of Prostate Cancer
48. Convenient Retinoid X Receptor Binding Assay Based on Fluorescence Change of the Antagonist NEt-C343.
49. Discovery of a "Gatekeeper" Antagonist that Blocks Entry Pathway to Retinoid X Receptors (RXRs) without Allosteric Ligand Inhibition in Permissive RXR Heterodimers.
50. Retinoid X Receptor Antagonists
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