315 results on '"Kireev, Dmitri"'
Search Results
2. Structural basis of paralog-specific KDM2A/B nucleosome recognition
3. Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors
4. A simulation model of heterochromatin formation at submolecular detail
5. Reprogramming CBX8-PRC1 function with a positive allosteric modulator
6. A chemical probe targeting the PWWP domain alters NSD2 nucleolar localization
7. Discovery of Novel Macrocyclic MERTK/AXL Dual Inhibitors
8. UNC5293, a potent, orally available and highly MERTK-selective inhibitor
9. The MERTK/FLT3 inhibitor MRX-2843 overcomes resistance-conferring FLT3 mutations in acute myeloid leukemia
10. Efforts toward discovering inhibitors of the SYK SH2–FCER1γ interaction as potential Alzheimer’s disease chemical probes and therapeutics
11. MERTK activation drives osimertinib resistance in EGFR-mutant non-small cell lung cancer
12. The entropic lock and key of the histone code
13. Discovery and Characterization of a Cellular Potent Positive Allosteric Modulator of the Polycomb Repressive Complex 1 Chromodomain, CBX7
14. Identification of Cosalane as an Inhibitor of Human and Murine CC–Chemokine Receptor 7 Signaling via a High-Throughput Screen
15. Machine Learning-driven Fragment-based Discovery of CIB1-directed Anti-Tumor Agents by FRASE-bot
16. Use of Protein Kinase–Focused Compound Libraries for the Discovery of New Inositol Phosphate Kinase Inhibitors
17. Application of Integrated Drug Screening/Kinome Analysis to Identify Inhibitors of Gemcitabine-Resistant Pancreatic Cancer Cell Growth
18. Supplementary Figure 3 from UNC569, a Novel Small-Molecule Mer Inhibitor with Efficacy against Acute Lymphoblastic Leukemia In Vitro and In Vivo
19. Supplementary Figure 2 from UNC569, a Novel Small-Molecule Mer Inhibitor with Efficacy against Acute Lymphoblastic Leukemia In Vitro and In Vivo
20. Supplementary Figure 4 from UNC569, a Novel Small-Molecule Mer Inhibitor with Efficacy against Acute Lymphoblastic Leukemia In Vitro and In Vivo
21. Supplementary Figure 1 from UNC569, a Novel Small-Molecule Mer Inhibitor with Efficacy against Acute Lymphoblastic Leukemia In Vitro and In Vivo
22. Data from UNC569, a Novel Small-Molecule Mer Inhibitor with Efficacy against Acute Lymphoblastic Leukemia In Vitro and In Vivo
23. Supplementary Figure 5 from UNC569, a Novel Small-Molecule Mer Inhibitor with Efficacy against Acute Lymphoblastic Leukemia In Vitro and In Vivo
24. Relationship between lysine methyltransferase levels and heterochromatin gene repression in living cells and in silico
25. PROTAC Linkerology Leads to an Optimized Bivalent Chemical Degrader of Polycomb Repressive Complex 2 (PRC2) Components
26. Dynamics of heterochromatin formation at submolecular resolution
27. Discovery of selective activators of PRC2 mutant EED-I363M
28. Development of a high-throughput TR-FRET screening assay for a fast-cycling KRAS mutant
29. Development of a High-Throughput Screening Assay to Identify Inhibitors of the Lipid Kinase PIP5K1C
30. Enzymatic Macrolactamization of mRNA Display Libraries for Inhibitor Selection
31. UNC1062, a new and potent Mer inhibitor
32. Inhibitors of Streptococcus pneumoniae Surface Endonuclease EndA Discovered by High-Throughput Screening Using a PicoGreen Fluorescence Assay
33. Multivalent DNA and nucleosome acidic patch interactions specify VRK1 mitotic localization and activity
34. List of Contributors
35. Structure-Based Virtual Screening of Commercially Available Compound Libraries
36. Computational Chemical Biology of Methyllysine Histone Effectors
37. Use of AD Informer Set compounds to explore validity of novel targets in Alzheimer's disease pathology
38. AD Informer Set: Chemical tools to facilitate Alzheimer's disease drug discovery
39. Combining Pharmacophore Models Derived from DNA-Encoded Chemical Libraries with Structure-Based Exploration to Predict Tankyrase 1 Inhibitors
40. Generation of the AD Informer Set: Chemical tools to facilitate Alzheimer’s disease drug discovery
41. A chemical probe targeting the PWWP domain alters NSD2 nucleolar localization
42. Enzymatic Macrolactamization of mRNA Display Libraries for Inhibitor Selection.
43. Screening for Inhibitors of Low-Affinity Epigenetic Peptide-Protein Interactions: An AlphaScreen™-Based Assay for Antagonists of Methyl-Lysine Binding Proteins
44. Discovery and Development of Cyclic Peptide Inhibitors of CIB1
45. AD Informer Set: Chemical tools to facilitate Alzheimer’s disease drug discovery
46. Correction to “A Focused DNA-Encoded Chemical Library for the Discovery of Inhibitors of NAD+-Dependent Enzymes”
47. Integrating DNA-encoded chemical libraries with virtual combinatorial library screening: Optimizing a PARP10 inhibitor
48. Pharmacological targeting of a PWWP domain demonstrates cooperative control of NSD2 localization
49. REPROGRAMMING CBX8-PRC1 FUNCTION WITH A POSITIVE ALLOSTERIC MODULATOR
50. A CoMFA Study of Enantiomeric Organophoshorus Inhibitors of Acetylcholinesterase
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