49 results on '"Lebel, Lorraine"'
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2. Inhibition of the striatum-enriched phosphodiesterase PDE10A: A novel approach to the treatment of psychosis
3. Small-molecule phosphodiesterase probes: discovery of potent and selective CNS-penetrable quinazoline inhibitors of PDE1
4. The discovery of a structurally novel class of inhibitors of the type 1 glycine transporter
5. Synthesis and SAR studies of 1,4-diazabicyclo[3.2.2]nonane phenyl carbamates – subtype selective, high affinity α7 nicotinic acetylcholine receptor agonists
6. Deconstructing cytisine: The syntheses of (±)-cyfusine and (±)-cyclopropylcyfusine, fused ring analogs of cytisine
7. Use of Structure-Based Design to Discover a Potent, Selective, In Vivo Active Phosphodiesterase 10A Inhibitor Lead Series for the Treatment of Schizophrenia
8. Corrigendum to “The discovery of a structurally novel class of inhibitors of the type 1glycine transporter” [Bioorg. Med. Chem. Lett. 19 (2009) 2974]
9. Discovery of a Series of 6,7-Dimethoxy-4-pyrrolidylquinazoline PDE10A Inhibitors
10. 3,5-Bicyclic aryl piperidines: A novel class of α4β2 neuronal nicotinic receptor partial agonists for smoking cessation
11. In pursuit of α4β2 nicotinic receptor partial agonists for smoking cessation: Carbon analogs of (−)-cytisine
12. Varenicline: An α4β2 Nicotinic Receptor Partial Agonist for Smoking Cessation
13. [3H]-(R)-NPTS, a radioligand for the type 1 glycine transporter
14. Ziprasidone: a novel antipsychotic agent with a unique human receptor binding profile
15. 5-cyano-1-[3-(N-methylpyrrolidin-2R-ylmethyl)indol-5-yl] benzimidazole (CP-161,242): A potent, centrally active 5-HT1D receptor agonist and benzodiazepine partial agonist
16. Dopamine uptake inhibitory activity of novel tryptamine 5‐HT1 receptor ligands
17. 5-[(3-Nitropyrid-2-yl)amino]indoles: Novel Serotonin Agonists with Selectivity for the 5-HT1D Receptor. Variation of the C3 Substituent on the Indole Template Leads to Increased 5-HT1D Receptor Selectivity
18. Synthesis and serotonergic pharmacology of the enantiomers of 3-[(N-methylpyrrolidin-2-yl)methyl]-5-methoxy-1H-indole: discovery of stereogenic differentiation in the aminoethyl side chain of the neurotransmitter serotonin
19. 1-(2-Aminoethyl)-3-methyl-8,9-dihydropyrano[3,2-e]indole: a rotationally restricted phenolic analog of the neurotransmitter serotonin and agonist selective for serotonin (5-HT2-type) receptors
20. Characterization of [3H]CP-96,501 as a Selective Radioligand for the Serotonin 5-HT1BReceptor: Binding Studies in Rat Brain Membranes
21. Binding studies with the 5-HT1B receptor agonist [3H]CP-96,501 in brain tissues
22. Binding and uptake studies with [3H]CP-93, 129, a radiolabeled selective 5-HT1B receptor ligand
23. Synthesis of 5-(2,3-ditritiopropoxy)-3-(1,2,5,6-tetrahydropyrid-4-yl)indole ([3H]CP-96,501): A selective ligand for the serotonin (5-HT1B) receptor
24. Structure-activity relationship of quinazolinedione inhibitors of calcium-independent phosphodiesterase
25. Nicotinamide ethers: novel inhibitors of calcium-independent phosphodiesterase and [3H]rolipram binding
26. Calcium-independent phosphodiesterase inhibitors as putative antidepressants: [3-(bicycloalkyloxy)-4-methoxyphenyl-2-imidazolidinones
27. 4-Amino[1,2,4]triazolo[4,3-a]quinoxalines. A novel class of potent adenosine receptor antagonists and potential rapid-onset antidepressants
28. 3-(1,2,5,6-Tetrahydropyrid-4-yl)pyrrolo[3,2-b]pyrid-5-one: a potent and selective serotonin (5-HT1*) agonist and rotationally restricted phenolic analog of 5-methoxy-3-(1,2,5,6-tetrahydropyrid-4-yl)indole
29. Effects of novel catechol ether imidazolidinones on calcium‐independent phosphodiesterase activity, [3H]rolipram binding, and reserpine‐induced hypothermia in mice
30. Dopamine uptake inhibitory activity of novel tryptamine 5-HT1 receptor ligands.
31. Synthesis of 5-(2,3-ditritiopropoxy)-3-(1,2,5,6-tetrahydropyrid-4-yl)indole ([3H]CP-96,501): A selective ligand for the serotonin (5-HT1B) receptor.
32. Characterization of [3H]CP-96,501 as a Selective Radioligand for the Serotonin 5-HT1B Receptor: Binding Studies in Rat Brain Membranes.
33. Binding studies with the 5-HT1B receptor agonist [3H]CP-96,501 in brain tissues.
34. Binding and uptake studies with [3H]CP-93, 129, a radiolabeled selective 5-HT1B receptor ligand.
35. Effects of novel catechol ether imidazolidinones on calcium-independent phosphodiesterase activity, [3H]rolipram binding, and reserpine-induced hypothermia in mice.
36. Enhancement of benzodiazepine binding by methaqualone and related quinazolinones.
37. Biochemical evidence for a new benzodiazepine receptor antagonist.
38. Varenicline:? An a4ß2 Nicotinic ReceptorPartial Agonist for Smoking Cessation
39. Sertraline potently displaces (+)-[3H]3-PPP binding to σ sites in rat brain
40. (+)-[3H]3-(3-hydroxyphenyl)-N-(1-propyl)-piperidine binding to σ receptors in mouse brain in vivo
41. Sertraline, a selective inhibitor of serotonin uptake, induces subsensitivity of β-adrenoceptor system of rat brain
42. 5-cyano-1-[3-(N-methylpyrrolidin-2R-ylmethyl)indol-5-yl] benzimidazole (CP-161,242): A potent, centrally active 5-HT 1D receptor agonist and benzodiazepine partial agonist
43. Contrasting effects of ethyl β-carboline-3-carboxylate (βCCE) and diazepam on cerebellar cyclic GMP content and antagonism of both effects by Ro 15-1788, a specific benzodiazepine receptor blocker
44. [3H]-(R)-NPTS, a radioligand for the type 1 glycine transporter
45. Synthesis and SAR studies of 1,4-diazabicyclo[3.2.2]nonane phenyl carbamates--subtype selective, high affinity alpha7 nicotinic acetylcholine receptor agonists.
46. Discovery of a series of 6,7-dimethoxy-4-pyrrolidylquinazoline PDE10A inhibitors.
47. 3,5-Bicyclic aryl piperidines: a novel class of alpha4beta2 neuronal nicotinic receptor partial agonists for smoking cessation.
48. In pursuit of alpha4beta2 nicotinic receptor partial agonists for smoking cessation: carbon analogs of (-)-cytisine.
49. Varenicline: an alpha4beta2 nicotinic receptor partial agonist for smoking cessation.
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