109 results on '"Mistry, Shailesh N."'
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2. Assessment of the potential of novel and classical opioids to induce respiratory depression in mice
3. Design, Synthesis, and Application of Fluorescent Ligands Targeting the Intracellular Allosteric Binding Site of the CXC Chemokine Receptor 2
4. Potent dual inhibitors of Plasmodium falciparum M1 and M17 aminopeptidases through optimization of S1 pocket interactions
5. M 1 muscarinic receptor activation reduces the molecular pathology and slows the progression of prion-mediated neurodegenerative disease
6. Development of fluorescent peptide G protein‐coupled receptor activation biosensors for NanoBRET characterization of intracellular allosteric modulators
7. Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H1 Receptor
8. Development of fluorescent peptide G Protein Coupled Receptor activation biosensors for NanoBRET characterisation of intracellular allosteric modulators
9. M1 muscarinic receptor activation reduces the molecular pathology and slows the progression of prion-mediated neurodegenerative disease.
10. Activation of M1 muscarinic receptors reduce pathology and slow progression of neurodegenerative disease
11. Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H1 Receptor.
12. Hit Identification of New Potent PqsR Antagonists as Inhibitors of Quorum Sensing in Planktonic and Biofilm Grown Pseudomonas aeruginosa
13. 27th Annual GP2A Medicinal Chemistry Conference
14. Structure–Kinetic Profiling of Haloperidol Analogues at the Human Dopamine D2 Receptor
15. Novel selective ?1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease
16. Positive allosteric modulation of the muscarinic M1 receptor improves efficacy of antipsychotics in mouse glutamatergic deficit models of behavior
17. Assessment of the Molecular Mechanisms of Action of Novel 4-Phenylpyridine-2-One and 6-Phenylpyrimidin-4-One Allosteric Modulators at the M1 Muscarinic Acetylcholine Receptors
18. A Thieno[2,3-d]pyrimidine Scaffold Is a Novel Negative Allosteric Modulator of the Dopamine D2 Receptor
19. The composite influence of the imidazolone moiety of CGP 12177 on its affinity and efficacy at the two conformations of the human β1-adrenoceptor
20. The effect of the N-alkyl moiety on the interaction of pindolol analogues with the two agonist conformations of the human β1-adrenoceptor
21. 4-Phenylpyridin-2-one Derivatives: A Novel Class of Positive Allosteric Modulator of the M1 Muscarinic Acetylcholine Receptor
22. Novel selective β 1 ‐adrenoceptor antagonists for concomitant cardiovascular and respiratory disease
23. Structure–activity study of N-((trans)-4-(2-(7-cyano-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)cyclohexyl)-1H-indole-2-carboxamide (SB269652), a bitopic ligand that acts as a negative allosteric modulator of the dopamine D2 receptor
24. Molecular determinants of allosteric modulation at the M1 muscarinic acetylcholine receptor
25. Positive Allosteric Modulation of the Muscarinic M1Receptor Improves Efficacy of Antipsychotics in Mouse Glutamatergic Deficit Models of Behavior
26. GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors
27. Novel Fused Arylpyrimidinone Based Allosteric Modulators of the M1 Muscarinic Acetylcholine Receptor
28. 4-Phenylpyridin-2-one Derivatives: A Novel Class of Positive Allosteric Modulator of the M1 Muscarinic Acetylcholine Receptor
29. Synthesis and in vitro and in vivo characterization of highly ?1-Selective ?-Adrenoceptor partial agonists
30. A Thieno[2,3-d]pyrimidine Scaffold Is a Novel Negative Allosteric Modulator of the Dopamine D2Receptor
31. In vitro and in vivo analysis of a novel highly selective β1-adrenoceptor partial agonist
32. Discovery of a Novel Class of Negative Allosteric Modulator of the Dopamine D2 Receptor Through Fragmentation of a Bitopic Ligand
33. Screening the Medicines for Malaria Venture "Malaria Box" against the Plasmodium falciparum Aminopeptidases, M1, M17 and M18
34. Mechanistic Insights into Allosteric Structure-Function Relationships at the M1 Muscarinic Acetylcholine Receptor
35. Two-Pronged Attack: Dual Inhibition of Plasmodium falciparum M1 and M17 Metalloaminopeptidases by a Novel Series of Hydroxamic Acid-Based Inhibitors
36. GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors.
37. Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease.
38. Triphenylphosphonium Anhydride Trifluoromethanesulfonate
39. Assessment of the Molecular Mechanisms of Action of Novel 4-Phenylpyridine-2-One and 6-Phenylpyrimidin-4-One Allosteric Modulators at the M1Muscarinic Acetylcholine Receptors
40. Synthesis and Pharmacological Profiling of Analogues of Benzyl Quinolone Carboxylic Acid (BQCA) as Allosteric Modulators of the M1 Muscarinic Receptor
41. Synthesis and in Vitro and in Vivo Characterization of Highly β1-Selective β-Adrenoceptor Partial Agonists
42. 4-Phenylpyridin-2-one Derivatives: A Novel Class of Positive Allosteric Modulator of the M1 Muscarinic Acetylcholine Receptor.
43. 4,5-Dihydro-1-[(1S)-1-(hydroxymethyl)-2,2-dimethylpropyl]-3-(2,4,6-trimethylphenyl)-1H-imidazolium Hexafluorophosphate
44. Synthesis and Characterization of High-Affinity 4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene-Labeled Fluorescent Ligands for Human β-Adrenoceptors
45. Triphenylphosphonium Anhydride Trifluoromethanesulfonate
46. Discovery of a Novel Class of Negative Allosteric Modulator of the Dopamine D2 Receptor Through Fragmentation of a Bitopic Ligand.
47. Two-Pronged Attack: Dual Inhibitionof Plasmodium falciparumM1 and M17Metalloaminopeptidasesby a Novel Series of Hydroxamic Acid-Based Inhibitors.
48. Synthesisand Pharmacological Profiling of Analoguesof Benzyl Quinolone Carboxylic Acid (BQCA) as Allosteric Modulatorsof the M1Muscarinic Receptor.
49. Synthesisand in Vitro and in Vivo Characterizationof Highly β1-Selective β-AdrenoceptorPartial Agonists.
50. Synthesis and Characterization of High-Affinity 4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene-Labeled Fluorescent Ligands for Human β-Adrenoceptors.
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