249 results on '"Picaud, Sarah"'
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2. Histone H4K16ac Binding Function of the Triple PHD Finger Cassette of MLL4
3. DNA damage remodels the MITF interactome to increase melanoma genomic instability
4. BRAF/MAPK and GSK3 signaling converges to control MITF nuclear export
5. The C-terminal extension landscape of naturally presented HLA-I ligands
6. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
7. Development and preclinical validation of a novel covalent ubiquitin receptor Rpn13 degrader in multiple myeloma
8. Histone H4K16ac binding function of the triple PHD finger cassette of MLL4
9. DNA damage-induced interaction between a lineage addiction oncogenic transcription factor and the MRN complex shapes a tissue-specific DNA Damage Response and cancer predisposition
10. Supplemental Methods and References from Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy
11. Supplementary Tables S1-S8 from Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy
12. Data from Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy
13. Supplemental Figures S1-S6 from Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy
14. Front Cover: Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain (ChemMedChem 20/2022)
15. Discovery of Benzo[ d ]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain
16. RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain
17. Small molecule inhibitors reveal an indispensable scaffolding role of RIPK2 in NOD2 signaling
18. Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family
19. Acetylation reprograms MITF target selectivity
20. Discovery of Novel BRD4 Ligand Scaffolds by Automated Navigation of the Fragment Chemical Space
21. The structure of nontypeable Haemophilus influenzae SapA in a closed conformation reveals a constricted ligand-binding cavity and a novel RNA binding motif
22. Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain.
23. Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain
24. Probing BRD Inhibition Substituent Effects in Bulky Analogues of (+)‐JQ1
25. Structural basis of fumarate hydratase deficiency
26. BRD4 methylation by the methyltransferase SETD6 regulates selective transcription to control mRNA translation
27. Supplementary Figures 1 and 2 from Identification of a PGXPP degron motif in dishevelled and structural basis for its binding to the E3 ligase KLHL12
28. Probing BRD Inhibition Substituent Effects in Bulky Analogues of (+)‐JQ1
29. Identification of a PGXPP degron motif in dishevelled and structural basis for its binding to the E3 ligase KLHL12
30. Controlling Intramolecular Interactions in the Design of Selective, High-Affinity, Ligands for the CREBBP Bromodomain
31. Selective inhibition of BET bromodomains
32. Synthesis and Biological Investigation of (+)-JD1, an Organometallic BET Bromodomain Inhibitor
33. Cloning and expression of a hexose transporter gene expressed during the ripening of grape berry (1)
34. Interactome Rewiring Following Pharmacological Targeting of BET Bromodomains
35. Structural Basis for Recruitment of DAPK1 to the KLHL20 E3 Ligase
36. A Tail-Based Mechanism Drives Nucleosome Demethylation by the LSD2/NPAC Multimeric Complex
37. Interactome Rewiring Following Pharmacological Targeting of BET Bromodomains
38. Evaluation of linker length effects on a BET bromodomain probe
39. Structural basis for recruitment of DAPK1 to the KLHL20 E3 ligase
40. Nut Directs p300-Dependent, Genome-Wide H4 Hyperacetylation in Male Germ Cells
41. Small molecule inhibitors reveal an indispensable scaffolding role of RIPK 2 in NOD 2 signaling
42. A TFEB nuclear export signal integrates amino acid supply and glucose availability
43. Promiscuous targeting of bromodomains by bromosporine identifies BET proteins as master regulators of primary transcription response in leukemia
44. Citrullination-acetylation interplay guides E2F-1 activity during the inflammatory response
45. The C-terminal extension landscape of naturally presented HLA-I ligands
46. Structures of PGAM5 Provide Insight into Active Site Plasticity and Multimeric Assembly
47. MOB1 Mediated Phospho-recognition in the Core Mammalian Hippo Pathway
48. Selective targeting of the BRG/PB1 bromodomains impairs embryonic and trophoblast stem cell maintenance
49. Multivalent Histone and DNA Engagement by a PHD/BRD/PWWP Triple Reader Cassette Recruits ZMYND8 to K14ac-Rich Chromatin
50. Synthesis and Biological Investigation of (+)-JD1, an Organometallic BET Bromodomain Inhibitor
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