17 results on '"Pinto, Donald J.P."'
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2. Structure based design of macrocyclic factor XIa inhibitors: Discovery of cyclic P1 linker moieties with improved oral bioavailability
3. Case History
4. Novel phenylalanine derived diamides as Factor XIa inhibitors
5. Terphenyl cyclooxygenase-2 (COX-2) inhibitors: Optimization of the central ring and o-biphenyl analogs
6. Structure-based design of inhibitors of coagulation factor XIa with novel P1 moieties
7. Orally bioavailable factor Xa inhibitors containing alpha-substituted gem-dimethyl P4 moieties
8. Phenyltriazolinones as potent factor Xa inhibitors
9. Structure–activity relationship and pharmacokinetic profile of 5-ketopyrazole factor Xa inhibitors
10. Structure–activity relationships of anthranilamide-based factor Xa inhibitors containing piperidinone and pyridinone P4 moieties
11. Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residues
12. Discovery of potent, efficacious, and orally bioavailable inhibitors of blood coagulation factor Xa with neutral P1 moieties
13. 1-[3-Aminobenzisoxazol-5′-yl]-3-trifluoromethyl-6-[2′-(3-(R)-hydroxy-N-pyrrolidinyl)methyl-[1,1′]-biphen-4-yl]-1,4,5,6-tetrahydropyrazolo-[3,4-c]-pyridin-7-one (BMS-740808) a highly potent, selective, efficacious, and orally bioavailable inhibitor of blood coagulation factor Xa
14. Chemistry and pharmacokinetics of diarylthiophenes and terphenyls as selective COX-2 inhibitors
15. Inhibition of cartilage degradation by isothiazoloquinolinones
16. A nitrone-based approach to the synthesis of cis-3-amido azetidinones
17. A convenient route to azetidine-2,3-diones and cis-3β-amido azetidinones
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