408 results on '"Tourwé, Dirk A."'
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2. Azepinone-Constrained Amino Acids in Peptide and Peptidomimetic Design
3. Development of potent and proteolytically stable human neuromedin U receptor agonists
4. Opening the amino acid toolbox for peptide‐based NTS2‐selective ligands as promising lead compounds for pain management
5. Synthesis and binding characteristics of [3H]neuromedin N, a NTS2 receptor ligand
6. Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist – Neurokinin-1 antagonist peptidomimetics
7. Preservation of hepatocellular functionality in cultures of primary rat hepatocytes upon exposure to 4-Me 2N-BAVAH, a hydroxamate-based HDAC-inhibitor
8. Azepinone-Constrained Amino Acids in Peptide and Peptidomimetic Design
9. Using conformational constraints at position 6 of Angiotensin II to generate compounds with enhanced AT2R selectivity and proteolytic stability
10. Influence of ring substitution on the conformation and β-turn mimicry of 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one peptide mimetics
11. Identification of Dmt-D-Lys-Phe-Phe-OH as a highly antinociceptive tetrapeptide metabolite of the opioid-neurotensin hybrid peptide PK20
12. PEGylation, increasing specific activity and multiple dosing as strategies to improve the risk-benefit profile of targeted radionuclide therapy with 177Lu-DOTA-bombesin analogues
13. Synergetic effects of DNA demethylation and histone deacetylase inhibition in primary rat hepatocytes
14. New tetracyclic tetrahydro-β-carbolines as tryptophan-derived peptidomimetics
15. Carbohydrated [99mTc(CO)3](NαHis)Ac-Bombesin(7–14) analogs
16. Screening of amide analogues of Trichostatin A in cultures of primary rat hepatocytes: search for potent and safe HDAC inhibitors
17. A stable neurotensin-based radiopharmaceutical for targeted imaging and therapy of neurotensin receptor-positive tumours
18. Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
19. Maillard Glycation of Peptides Containing the (N αHis)Ac Chelator for 99mTc(CO)3 Labeling
20. Synthesis of 4-amino-1,2,4,5-tetrahydro-2-benzazepine-3-ones and Study of their β-turn Inducing Properties
21. An Asymmetric Synthesis of (R)- and (S)-o-cyano-phenylalanine Leading to Chiral Constrained Phenylalanine Dipeptide Mimetics
22. Chemical and biological characterization of new Re(CO) 3/[ 99mTc](CO) 3 bombesin analogues
23. Derivatization of 1-phenyl substituted 4-amino-2-benzazepin-3-ones: evaluation of Pd-catalyzed coupling reactions
24. Synthesis of 4-amino-3-oxo-tetrahydroazepino[3,4- b]indoles: new conformationally constrained Trp analogs
25. Neuromedin U and Structural Analogs: An Overview of their Structure, Function and Selectivity
26. Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal Structure
27. [3H]IVDE77, a novel radioligand with high affinity and selectivity for the insulin-regulated aminopeptidase
28. Cyclic Somatostatins containing α-benzyl-o-AMPA as a cis peptide bond mimic
29. Double-stabilized neurotensin analogues as potential radiopharmaceuticals for NTR-positive tumors
30. Aspects of Peptidomimetics
31. Synthesis and binding properties of endomorphin-2analogs containing α-hydroxymethyl amino acids
32. Synthesis and binding properties of endomorphin-2 analogs containing α-hydroxymethyl amino acids
33. Angiotensin IV displays only low affinity for native insulin-regulated aminopeptidase (IRAP)
34. Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure–Activity Relationship Studies
35. Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia
36. α-Bn-o-AMPA as a cis peptide bond mimic in somatostatin analogues
37. Glycation Methods for Bombesin Analogs Containing the (NαHis)Ac chelator for 99mTc(CO)3 Radiolabeling
38. Somatostatin analogues containing o-aminomethylphenylacetic acid as a bridge unit
39. New methods for solid phase peptide synthesis of transitionstate analog inhibitors of HIV-1 protease and DPP-IV
40. Conformation-directed design of cyclic somatostatins containing a βVI-turn mimetic
41. Maillard Glycation of Peptides Containing the (NαHis)Ac Chelator for 99mTc(CO)3 Labeling
42. CB&DD Editorial Advisory Board (fourth in series)
43. Comparison of the separation efficiencies of Chirobiotic T and TAG columns in the separation of unusual amino acids
44. Direct and indirect high-performance liquid chromatographic enantioseparation of β-amino acids
45. Biological Consequences of the Incorporation of Amphiphilic Amino Acids into Opioid Peptide Sequences
46. A versatile synthesis of 2-substituted 4-amino-1,2,4,5-tetrahydro-2-benzazepine-3-ones
47. Side reactions in the preparation of 1,2,3,4-tetrahydro-β-carboline-3-carboxylic acid
48. In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera
49. Trifluoromethylated Proline Surrogates as Part of “Pro–Pro” Turn‐Inducing Templates
50. Synthesis of the diastereomers of β-Me-Tyr and β-Me-Phe and their effect on the biological properties of the delta opioid receptor antagonist TIPP
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