30 results on '"Zhu, Juliang"'
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2. Design, Synthesis, and SAR of C-3 Benzoic Acid, C-17 Triterpenoid Derivatives. Identification of the HIV-1 Maturation Inhibitor 4-((1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-3a-((2-(1,1-Dioxidothiomorpholino)ethyl)amino)-5a,5b,8,8,11a-pentamethyl-1-(prop-1-en-2-yl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysen-9-yl)benzoic Acid (GSK3532795, BMS-955176)
3. Bioactivation of cyclopropyl rings by P450: an observation encountered during the optimisation of a series of hepatitis C virus NS5B inhibitors
4. Improving Metabolic Stability with Deuterium: The Discovery of BMT-052, a Pan-genotypic HCV NS5B Polymerase Inhibitor
5. The discovery of a pan-genotypic, primer grip inhibitor of HCV NS5B polymerase
6. Identification of 1-{2-[4-chloro-1′-(2,2-dimethylpropyl)-7-hydroxy-1,2-dihydrospiro[indole-3,4′-piperidine]-1-yl]phenyl}-3-{5-chloro-[1,3]thiazolo[5,4-b]pyridin-2-yl}urea, a potent, efficacious and orally bioavailable P2Y1 antagonist as an antiplatelet agent
7. An Efficient Scale-Up Synthesis of BMS-520, a Potent and Selective Isoxazole-Containing S1P1 Receptor Agonist
8. Discovery of BMS-955176, a Second Generation HIV-1 Maturation Inhibitor with Broad Spectrum Antiviral Activity
9. Discovery and Preclinical Evaluation of BMS-711939, an Oxybenzylglycine Based PPARα Selective Agonist
10. An effective procedure for the acylation of azaindoles at C-3
11. Hepatitis C Virus NS5A Replication Complex Inhibitors: The Discovery of Daclatasvir
12. Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment 6. Preclinical and Human Pharmacokinetic Profiling of BMS-663749, a Phosphonooxymethyl Prodrug of the HIV-1 Attachment Inhibitor 2-(4-Benzoyl-1-piperazinyl)-1-(4,7-dimethoxy-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-oxoethanone (BMS-488043)
13. An Effective Procedure for the Preparation of 3-Substituted 4- or 6-Azaindoles from ortho-Methylnitropyridines.
14. An effective procedure for the preparation of 3-substituted-4- or 6-azaindoles from ortho-methyl nitro pyridines
15. Synthesis of Substituted Aryl Amidines from Aminoacetonitriles.
16. A One‐Pot Synthesis of Nitrogen‐Containing Heteroaryl α‐Keto Amides from Heteroaryl Halides.
17. Malononitrile as a Carbonyl Synthon: A One‐Pot Preparation of Heteroaryl Amide via a SNAr‐Oxidation—Displacement Strategy.
18. Malononitrile as a carbonyl synthon: a one-pot preparation of heteroaryl amide via a S N Ar-oxidation–displacement strategy
19. An Effective Procedure for the Acylation of Azaindoles at C‐3.
20. (+)-Dinapsoline: An Efficient Synthesis and Pharmacological Profile of a Novel Dopamine Agonist
21. Hepatitis C Virus NS5A Replication Complex Inhibitors:The Discovery of Daclatasvir.
22. Synthesis of substituted aryl amidines from aminoacetonitriles
23. A one-pot synthesis of nitrogen-containing heteroaryl α-keto amides from heteroaryl halides
24. Malononitrile as a carbonyl synthon: a one-pot preparation of heteroaryl amide via a SNAr-oxidation–displacement strategy
25. Anti-HIV-1 activity and cellular pharmacology of various analogs of gossypol
26. Inhibitors of Human ImmunodeficiencyVirus Type 1(HIV-1) Attachment 6. Preclinical and Human Pharmacokinetic Profilingof BMS-663749, a Phosphonooxymethyl Prodrug of the HIV-1 AttachmentInhibitor...
27. Malononitrile as a carbonyl synthon: a one-pot preparation of heteroaryl amide via a SNAr-oxidation–displacement strategy
28. Identification of 1-{2-[4-chloro-1′-(2,2-dimethylpropyl)-7-hydroxy-1,2-dihydrospiro[indole-3,4′-piperidine]-1-yl]phenyl}-3-{5-chloro-[1,3]thiazolo[5,4-b]pyridin-2-yl}urea, a potent, efficacious and orally bioavailable P2Y1 antagonist as an antiplatelet agent.
29. Bioactivation of cyclopropyl rings by P450: an observation encountered during the optimisation of a series of hepatitis C virus NS5B inhibitors.
30. Design, Synthesis, and SAR of C-3 Benzoic Acid, C-17 Triterpenoid Derivatives. Identification of the HIV-1 Maturation Inhibitor 4-((1 R,3a S,5a R,5b R,7a R,11a S,11b R,13a R,13b R)-3a-((2-(1,1-Dioxidothiomorpholino)ethyl)amino)-5a,5b,8,8,11a-pentamethyl-1-(prop-1-en-2-yl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1 H-cyclopenta[ a]chrysen-9-yl)benzoic Acid (GSK3532795, BMS-955176).
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