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1. Assessment In vitro and In silico of the Activity of Thiadiazines as NorA Efflux Pump Inhibitors

2. List of contributors

3. New drug discovery and development

4. Preclinical data on morpholine (3,5-di-tertbutyl-4-hydroxyphenyl) methanone induced anxiolysis

7. Larvicidal activity, enzyme inhibitory effect, and molecular docking by essential oil, hydrolate, aqueous extract, and major compounds from the leaves of Eugenia uniflora against Aedes aegypti

9. Antiviral agents against flaviviruses

10. A consensus reverse docking approach for identification of a competitive inhibitor of acetyltransferase enhanced intracellular survival protein from Mycobacterium tuberculosis

12. The Medicinal Chemistry of Zika Virus

14. PI3K Signaling Pathways as a Molecular Target for Glioblastoma Multiforme

19. An electrochemical biosensor based on Hairpin-DNA modified gold electrode for detection of DNA damage by a hybrid cancer drug intercalation

20. Potentiating‐antibiotic activity and absorption, distribution, metabolism, excretion and toxicity properties (ADMET) analysis of synthetic thiadiazines against multi‐drug resistant (MDR) strains.

22. Potentiating‐antibiotic activity and absorption, distribution, metabolism, excretion and toxicity properties (ADMET) analysis of synthetic thiadiazines against multi‐drug resistant (MDR) strains

36. Medicinal Chemistry of Inhibitors Targeting Resistant Bacteria

37. Oviposition deterrence, larvicidal activity and docking of β-germacrene-D-4-ol obtained from leaves of Piper corcovadensis (Piperaceae) against Aedes aegypti

40. In vitro antitumor activity of dialkylamine-1,4-naphthoquinones toward human glioblastoma multiforme cells

42. Dual quinoline-hybrid compounds with antimalarial activity against Plasmodium falciparum parasites

48. Druggable targets from coronaviruses for designing new antiviral drugs

49. Contributors

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