488 results on '"van der Stelt, Mario"'
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2. Structural basis of selective cannabinoid CB2 receptor activation
3. Dual allosteric and orthosteric pharmacology of synthetic analog cannabidiol-dimethylheptyl, but not cannabidiol, on the cannabinoid CB2 receptor
4. THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Enzymes
5. Oxygenation of Anandamide by Lipoxygenases
6. Fluorescence-Based NAPE-PLD Activity Assay
7. Cellular Assay to Study β-Arrestin Recruitment by the Cannabinoid Receptors 1 and 2
8. Multi-parameter optimization: Development of a morpholin-3-one derivative with an improved kinetic profile for imaging monoacylglycerol lipase in the brain
9. P2X7 receptor‐dependent increase in endocannabinoid 2‐arachidonoyl glycerol production by neuronal cells in culture: Dynamics and mechanism.
10. Discovery of a Cannabinoid CB2 Receptor Fluorescent Probe Based on a Pyridin-2-yl-benzyl-imidazolidine-2,4-dione Scaffold.
11. Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
12. Stress-induced modulation of endocannabinoid signaling leads to delayed strengthening of synaptic connectivity in the amygdala
13. Discovery of a Photoaffinity Probe that Captures the Active Conformation of the Cannabinoid CB2 Receptor.
14. Opportunities for Lipid-Based Probes in the Field of Immunology
15. PharmacoSTORM nanoscale pharmacology reveals cariprazine binding on Islands of Calleja granule cells
16. Biochemical and Cellular Characterization of the Function of Fluorophosphonate-Binding Hydrolase H (FphH) in Staphylococcus aureus Support a Role in Bacterial Stress Response
17. IMI European Lead Factory — democratizing access to high-throughput screening
18. Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice
19. Improving CLL Vγ9Vδ2-T–cell fitness for cellular therapy by ex vivo activation and ibrutinib
20. Disruption of tonic endocannabinoid signalling triggers cellular, behavioural and neuroendocrine responses consistent with a stress response.
21. Structural basis of selective cannabinoid CB2 receptor activation
22. A novel antifolate suppresses growth of FPGS-deficient cells and overcomes methotrexate resistance
23. Regulation of Adipose Tissue Metabolism by the Endocannabinoid System
24. Piperidine and octahydropyrano[3,4-c] pyridine scaffolds for drug-like molecular libraries of the European Lead Factory
25. Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474
26. Goods and bads of endocannabinoid system as a therapeutic target:Lessons learned after 30 years
27. Endocannabinoid turnover in GtoPdb v.2023.1
28. CB1 Cannabinoid Receptors and On-Demand Defense against Excitotoxicity
29. Chemical genetics strategy to profile kinase target engagement reveals role of FES in neutrophil phagocytosis
30. Inhibition of diacylglycerol lipase β modulates lipid and endocannabinoid levels in the ex vivo human placenta
31. Understanding and Targeting the Endocannabinoid System with Activity‐Based Protein Profiling
32. EFMC – Trends that Link Medicinal Chemistry and Chemical Biology to Translational Drug Discovery
33. Anandamide and other N-acylethanolamines: A class of signaling lipids with therapeutic opportunities
34. Chemical Proteomics Reveals Antibiotic Targets of Oxadiazolones in MRSA
35. 2-AG-Mediated Control of GABAergic Signaling Is Impaired in a Model of Epilepsy
36. Inhibitors of diacylglycerol lipases in neurodegenerative and metabolic disorders
37. Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition
38. EFMC - trends that link medicinal chemistry and chemical biology to translational drug discovery
39. Goods and bads of endocannabinoid system as a therapeutic target: Lessons learned after 30 years
40. Opportunities for Lipid-Based Probes in the Field of Immunology
41. Anti-neuroinflammatory effects of GPR55 antagonists in LPS-activated primary microglial cells
42. Cyclopentitol as a scaffold for a natural product-like compound library for drug discovery
43. Chemical Probes to Control and Visualize Lipid Metabolism in the Brain
44. Comparative Photoaffinity Profiling of Omega-3 Signaling Lipid Probes Reveals Prostaglandin Reductase 1 as a Metabolic Hub in Human Macrophages
45. Disruption of Tonic Endocannabinoid Signaling Triggers the Generation of a Stress Response
46. Live‐Cell Imaging of Sterculic Acid—a Naturally Occurring 1,2‐Cyclopropene Fatty Acid—by Bioorthogonal Reaction with Turn‐On Tetrazine‐Fluorophore Conjugates**
47. Evaluation of different drug classes on transient sciatic nerve injury–depressed marble burying in mice
48. Chemical tools to modulate 2‐arachidonoylglycerol biosynthesis
49. The endocannabinoid system and its therapeutic exploitation in multiple sclerosis: Clues for other neuroinflammatory diseases
50. Competitive ABPP of Serine Hydrolases: A Case Study on DAGL-Alpha
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