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Gallium(III)-Promoted Halocyclizations of 1,6-Diynes.

Authors :
Strom, Kyle R.
Impastato, Anna C.
Moy, Kenneth J.
Landreth, Adrian J.
Snyder, John K.
Source :
Organic Letters. May2015, Vol. 17 Issue 9, p2126-2129. 4p.
Publication Year :
2015

Abstract

Cyclization of 1,6-diynes promoted by stoichiometric Ga(III) halides produces vinyl halides in good to excellent yields. Under acidic conditions, initially formed iodocyclization products undergo in situ Friedel-Crafts cyclizations, giving access to iodoindenopyridines. Application of the vinyl halides in cross-coupling reactions has been explored, and mechanistic aspects of the cyclization are discussed. [ABSTRACT FROM AUTHOR]

Details

Language :
English
ISSN :
15237060
Volume :
17
Issue :
9
Database :
Academic Search Index
Journal :
Organic Letters
Publication Type :
Academic Journal
Accession number :
102476483
Full Text :
https://doi.org/10.1021/acs.orglett.5b00716