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Recent advances on the synthesis of acylindoles.
- Source :
-
Tetrahedron Letters: International Organ for the Rapid Publication of Preliminary Communications in Organic Chemistry . Aug2016, Vol. 57 Issue 35, p3892-3901. 10p. - Publication Year :
- 2016
-
Abstract
- Acylindoles are valuable chemicals widely found in natural products, pharmaceuticals, and biologically active compounds. They are also important synthetic building blocks for chemical transformation. Recent advances of acylindoles synthesis via acylation of indoles with diverse carbonyl sources ( N -alkylamines, aldehydes, α-oxocarboxylic acids, nitriles, olefins, CO, fluorinated acetic acids (salts), and diketones) are highly desirable methods. Moreover, intramolecular cyclization of aminoalkynes and enaminones also provided highly efficient and atom-economical alternatives to the traditional methods. Herein, we summarize recent advances on the synthesis of acylindoles. [ABSTRACT FROM AUTHOR]
Details
- Language :
- English
- ISSN :
- 00404039
- Volume :
- 57
- Issue :
- 35
- Database :
- Academic Search Index
- Journal :
- Tetrahedron Letters: International Organ for the Rapid Publication of Preliminary Communications in Organic Chemistry
- Publication Type :
- Academic Journal
- Accession number :
- 117292236
- Full Text :
- https://doi.org/10.1016/j.tetlet.2016.07.063