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Antimicrobial activity of new benzazolyl N-sulfonyl amidines.
- Source :
-
Mendeleev Communications . Jul2021, Vol. 31 Issue 4, p495-497. 3p. - Publication Year :
- 2021
-
Abstract
- [Display omitted] The reactions of N -(benz[ d ]oxazol-2-yl)- or N -(benzo[ d ]-thiazol-2-yl)-substituted carbothioamides with sulfonyl azides proceed as replacement of thioxo substituent by the sulfonylimino group to afford the corresponding N' -sulfonylated amidines. Acetic acid thioamides react smoothly upon boiling in ethanol, while for thioamides of trifluoroacetic and benzoic acids heating to 80–90 °C was required. Among hybrid molecules thus prepared, bacteriostatic-, bactericidal- and fungistatic-active against S. aureus and C. albicans representatives were found. [ABSTRACT FROM AUTHOR]
Details
- Language :
- English
- ISSN :
- 09599436
- Volume :
- 31
- Issue :
- 4
- Database :
- Academic Search Index
- Journal :
- Mendeleev Communications
- Publication Type :
- Academic Journal
- Accession number :
- 152006054
- Full Text :
- https://doi.org/10.1016/j.mencom.2021.07.019