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A Novel One-Step Synthesis of 2-Substituted 6-Azaindoles from 3-Amino-4-picoline and Carboxylic Esters.
- Source :
-
Journal of Organic Chemistry . 8/5/2005, Vol. 70 Issue 16, p6512-6514. 3p. 2 Diagrams, 1 Chart. - Publication Year :
- 2005
-
Abstract
- Dilithiation of 3-amino-4-picoline (1) was achieved with sec-BuLi at room temperature. Condensation of the resulting dianion (2) with carboxylic esters afforded a wide range of 2-substituted 6-azaindoles in good yields. [ABSTRACT FROM AUTHOR]
- Subjects :
- *INDOLE
*ORGANONITROGEN compounds
*ORGANIC synthesis
*ESTERS
*CONDENSATION
Subjects
Details
- Language :
- English
- ISSN :
- 00223263
- Volume :
- 70
- Issue :
- 16
- Database :
- Academic Search Index
- Journal :
- Journal of Organic Chemistry
- Publication Type :
- Academic Journal
- Accession number :
- 17882294
- Full Text :
- https://doi.org/10.1021/jo0506480