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Highly Potent Inhibitors of TNF-α Production. Part 1: Discovery of Chemical Leads

Authors :
Matsui, Toshiaki
Kondo, Takashi
Nishita, Yoshitaka
Itadani, Satoshi
Nakatani, Shingo
Omawari, Nagashige
Sakai, Masaru
Nakazawa, Shuichi
Ogata, Akihito
Ohno, Hiroyuki
Obata, Takaaki
Nakai, Hisao
Toda, Masaaki
Source :
Bioorganic & Medicinal Chemistry Letters. Mar2002, Vol. 12 Issue 6, p903. 3p.
Publication Year :
2002

Abstract

The discovery of 2-acylamino-2-phenylethyl disodium phosphates and as structurally novel inhibitors of TNF-α production is reported. Structure–activity relationships (SARs) are also discussed. [Copyright &y& Elsevier]

Details

Language :
English
ISSN :
0960894X
Volume :
12
Issue :
6
Database :
Academic Search Index
Journal :
Bioorganic & Medicinal Chemistry Letters
Publication Type :
Academic Journal
Accession number :
7761376
Full Text :
https://doi.org/10.1016/S0960-894X(02)00036-7