Back to Search
Start Over
Synthesis and structure–activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists
- Source :
-
Bioorganic & Medicinal Chemistry Letters . Aug2012, Vol. 22 Issue 15, p4986-4989. 4p. - Publication Year :
- 2012
-
Abstract
- Abstract: Pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones were evaluated as corticotropin-releasing factor-1 receptor antagonists. The synthesis, SAR studies and pharmacokinetic evaluation of these analogs are described herein. [Copyright &y& Elsevier]
Details
- Language :
- English
- ISSN :
- 0960894X
- Volume :
- 22
- Issue :
- 15
- Database :
- Academic Search Index
- Journal :
- Bioorganic & Medicinal Chemistry Letters
- Publication Type :
- Academic Journal
- Accession number :
- 78036770
- Full Text :
- https://doi.org/10.1016/j.bmcl.2012.06.034