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Factor VIIa inhibitors: improved pharmacokinetic parameters.

Authors :
Kolesnikov A
Rai R
Young WB
Mordenti J
Liu L
Torkelson S
Shrader WD
Leahy EM
Hu H
Gjerstad E
Janc J
Katz BA
Sprengeler PA
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2006 Apr 15; Vol. 16 (8), pp. 2243-6. Date of Electronic Publication: 2006 Feb 07.
Publication Year :
2006

Abstract

Efforts to improve the potency and pharmacokinetic properties of small molecule factor VIIa inhibitors are described. Small structural modifications to existing leads allow the modulation of half-life and clearance, potentially making these compounds suitable candidates for drug development.

Details

Language :
English
ISSN :
0960-894X
Volume :
16
Issue :
8
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
16455251
Full Text :
https://doi.org/10.1016/j.bmcl.2006.01.037