Back to Search Start Over

Substituted coumarins as potent 5-lipoxygenase inhibitors.

Authors :
Grimm EL
Brideau C
Chauret N
Chan CC
Delorme D
Ducharme Y
Ethier D
Falgueyret JP
Friesen RW
Guay J
Hamel P
Riendeau D
Soucy-Breau C
Tagari P
Girard Y
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2006 May 01; Vol. 16 (9), pp. 2528-31. Date of Electronic Publication: 2006 Feb 07.
Publication Year :
2006

Abstract

Leukotriene biosynthesis inhibitors have potential as therapeutic agents for asthma and inflammatory diseases. A novel series of substituted coumarin derivatives has been synthesized and the structure-activity relationship was evaluated with respect to their ability to inhibit the formation of leukotrienes via the human 5-lipoxygenase enzyme.

Details

Language :
English
ISSN :
0960-894X
Volume :
16
Issue :
9
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
16464579
Full Text :
https://doi.org/10.1016/j.bmcl.2006.01.085