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Design and synthesis of beta-methoxyacrylate analogues via click chemistry and biological evaluations.

Authors :
Chen H
Taylor JL
Abrams SR
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2007 Apr 01; Vol. 17 (7), pp. 1979-83. Date of Electronic Publication: 2007 Jan 19.
Publication Year :
2007

Abstract

A library of potential antifungal triazole-modified beta-methoxyacrylate analogues was designed and synthesized via a Cu(I)-catalyzed 1,3-dipolar alkyne-azide coupling reaction or 'click chemistry'. Subsequent biological screening revealed that some compounds displayed low to moderate antifungal activity toward pathogenic fungi and low phytotoxicity.

Details

Language :
English
ISSN :
0960-894X
Volume :
17
Issue :
7
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
17300931
Full Text :
https://doi.org/10.1016/j.bmcl.2007.01.021