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Identification of potential and selective collagenase, gelatinase inhibitors from Crataegus pinnatifida.

Authors :
Moon HI
Kim TI
Cho HS
Kim EK
Source :
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2010 Feb 01; Vol. 20 (3), pp. 991-3. Date of Electronic Publication: 2009 Dec 22.
Publication Year :
2010

Abstract

Four oligomeric procyanidins were isolated from the MeOH extracts of the leaves of Crataegus pinnatifida (Rosaceae). Investigation of collagenase and gelatinase inhibitory natural components afforded four oligomeric procyanidins. Of these, 2 and 3 exhibited collagenase inhibitory activity (IC(50)) at a concentration of less than 1 microM, and 3 showed gelatinases A and B inhibitory activity (IC(50)) at 0.4 and 2.3 microM, respectively.<br /> (Copyright (c) 2009 Elsevier Ltd. All rights reserved.)

Details

Language :
English
ISSN :
1464-3405
Volume :
20
Issue :
3
Database :
MEDLINE
Journal :
Bioorganic & medicinal chemistry letters
Publication Type :
Academic Journal
Accession number :
20053563
Full Text :
https://doi.org/10.1016/j.bmcl.2009.12.059