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A protocol for amide bond formation with electron deficient amines and sterically hindered substrates.

Authors :
Due-Hansen ME
Pandey SK
Christiansen E
Andersen R
Hansen SVF
Ulven T
Source :
Organic & biomolecular chemistry [Org Biomol Chem] 2016 Jan 14; Vol. 14 (2), pp. 430-433.
Publication Year :
2016

Abstract

A protocol for amide coupling by in situ formation of acyl fluorides and reaction with amines at elevated temperature has been developed and found to be efficient for coupling of sterically hindered substrates and electron deficient amines where standard methods failed.

Details

Language :
English
ISSN :
1477-0539
Volume :
14
Issue :
2
Database :
MEDLINE
Journal :
Organic & biomolecular chemistry
Publication Type :
Academic Journal
Accession number :
26586516
Full Text :
https://doi.org/10.1039/c5ob02129d