Back to Search Start Over

Preparation of Stereodefined 2-(3-Oxoindolin-2-yl)-2-Arylacetonitriles via One-Pot Reaction of Indoles with Nitroalkenes.

Authors :
Aksenov AV
Aksenov DA
Aksenov NA
Aleksandrova EV
Rubin M
Source :
The Journal of organic chemistry [J Org Chem] 2019 Oct 04; Vol. 84 (19), pp. 12420-12429. Date of Electronic Publication: 2019 Sep 18.
Publication Year :
2019

Abstract

Recently discovered reactivity of nitrostyrenes in phosphorous acid to facilitate the diastereoselective [4 + 1]-cycloaddition of indoles in combination with unusual oxazoline ring cleavage and subsequent 1,2-alkyl shift afforded stereochemically defined 2-(3-oxoindolin-2-yl)-2-arylacetonitriles as sole products.

Details

Language :
English
ISSN :
1520-6904
Volume :
84
Issue :
19
Database :
MEDLINE
Journal :
The Journal of organic chemistry
Publication Type :
Academic Journal
Accession number :
31502836
Full Text :
https://doi.org/10.1021/acs.joc.9b01874