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Bicyclo[6.1.0]nonyne carboxylic acid for the production of stable molecular probes.

Authors :
Rady T
Mosser M
Nothisen M
Erb S
Dovgan I
Cianférani S
Wagner A
Chaubet G
Source :
RSC advances [RSC Adv] 2021 Nov 17; Vol. 11 (58), pp. 36777-36780. Date of Electronic Publication: 2021 Nov 17 (Print Publication: 2021).
Publication Year :
2021

Abstract

Bicyclo[6.1.0]non-4-yn-9-ylmethanol (BCN alcohol) is the most prominent strained-alkyne scaffold in chemical biology. Described herein is the synthesis of an oxidized analogue - BCN acid - whose facile functionalization via amide bond formation yields more stable derivatives than the classically encountered carbamates.<br />Competing Interests: There are no conflicts to declare.<br /> (This journal is © The Royal Society of Chemistry.)

Details

Language :
English
ISSN :
2046-2069
Volume :
11
Issue :
58
Database :
MEDLINE
Journal :
RSC advances
Publication Type :
Academic Journal
Accession number :
35494363
Full Text :
https://doi.org/10.1039/d1ra07905k