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Cysteine-responsive prodrug of the anti-cancer drug amonafide: fluorogenic adjuvant drug delivery with hydrogen sulfide (H 2 S).

Authors :
Mahato SK
Barman P
Badirujjaman M
Bhabak KP
Source :
Chemical communications (Cambridge, England) [Chem Commun (Camb)] 2023 Apr 18; Vol. 59 (32), pp. 4802-4805. Date of Electronic Publication: 2023 Apr 18.
Publication Year :
2023

Abstract

L-Cysteine (Cys)-responsive turn-on fluorogenic prodrug AM-ITC was developed for the adjuvant delivery of the anti-cancer drug amonafide and the gasotransmitter hydrogen sulfide (H <subscript>2</subscript> S) in aqueous and cellular media. Considering the cytoprotective roles of H <subscript>2</subscript> S, the present adjuvant strategy would be helpful in minimizing the anti-cancer drug-induced side-effects.

Details

Language :
English
ISSN :
1364-548X
Volume :
59
Issue :
32
Database :
MEDLINE
Journal :
Chemical communications (Cambridge, England)
Publication Type :
Academic Journal
Accession number :
37000594
Full Text :
https://doi.org/10.1039/d3cc00220a