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Enantioselective de novo synthesis of 14-hydroxy-6-oxomorphinans.

Authors :
Moore JC
Modell L
Glenn JR
Jones KD
Argent SP
Lane JR
Canals M
Lam HW
Source :
Chemical communications (Cambridge, England) [Chem Commun (Camb)] 2024 Jun 06; Vol. 60 (47), pp. 6007-6010. Date of Electronic Publication: 2024 Jun 06.
Publication Year :
2024

Abstract

The enantioselective de novo synthesis of pharmacologically important 14-hydroxy-6-oxomorphinans is described. 4,5-Desoxynaltrexone and 4,5-desoxynaloxone were prepared using this route and their biological activities against the opioid receptors were measured.

Details

Language :
English
ISSN :
1364-548X
Volume :
60
Issue :
47
Database :
MEDLINE
Journal :
Chemical communications (Cambridge, England)
Publication Type :
Academic Journal
Accession number :
38787679
Full Text :
https://doi.org/10.1039/d4cc01788a