Back to Search Start Over

A Facile Synthesis for Novel Loperamide Analogs as Potential μOpioid Receptor Agonists.

Authors :
Xiaofeng Bao
Duliang Liu
Yanyan Jin
Yao Yang
Source :
Molecules; Dec2012, Vol. 17 Issue 12, p14288-14297, 10p, 5 Diagrams, 2 Charts
Publication Year :
2012

Abstract

A facile synthesis for novel loperamide analogs as potential μ opioid receptors is described. The synthetic procedure for compound 5, which contains two 4-phenyl piperidine scaffolds, was optimized, and this compound was synthesized in excellent yield. We also describe a mild and highly efficient protocol for the synthesis of compounds 6 and 7. [ABSTRACT FROM AUTHOR]

Details

Language :
English
ISSN :
14203049
Volume :
17
Issue :
12
Database :
Complementary Index
Journal :
Molecules
Publication Type :
Academic Journal
Accession number :
84451551
Full Text :
https://doi.org/10.3390/molecules171214288