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A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs.

Authors :
Bhela, Irene Preet
Ranza, Alice
Balestrero, Federica Carolina
Serafini, Marta
Aprile, Silvio
Di Martino, Rita Maria Concetta
Condorelli, Fabrizio
Pirali, Tracey
Source :
Journal of Medicinal Chemistry; 11/24/2022, Vol. 65 Issue 22, p15282-15299, 18p
Publication Year :
2022

Details

Language :
English
ISSN :
00222623
Volume :
65
Issue :
22
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
160430205
Full Text :
https://doi.org/10.1021/acs.jmedchem.2c01218