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Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV‑1 Activities and Improved Oral Bioavailability.

Authors :
Xie, Xiong
Zheng, Yu-Gui
Chen, Huan
Li, Jian
Luo, Rong-Hua
Chen, Liang
Zheng, Chang-Bo
Zhang, Shurui
Peng, Panfeng
Ma, Dakota
Yang, Liu-Meng
Zheng, Yong-Tang
Liu, Hong
Wang, Jiang
Source :
Journal of Medicinal Chemistry; 12/22/2022, Vol. 65 Issue 24, p16526-16540, 15p
Publication Year :
2022

Details

Language :
English
ISSN :
00222623
Volume :
65
Issue :
24
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
160956349
Full Text :
https://doi.org/10.1021/acs.jmedchem.2c01383