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X‑ray Structure-Guided Discovery of a Potent Benzimidazole Glutaminyl Cyclase Inhibitor That Shows Activity in a Parkinson's Disease Mouse Model.

Authors :
Mou, Jun
Ning, Xiang-Li
Wang, Xin-Yue
Hou, Shu-Yan
Meng, Fan-Bo
Zhou, Cong
Wu, Jing-Wei
Li, Chunyan
Jia, Tao
Wu, Xiaoai
Wu, Yong
Chen, Yongping
Li, Guo-Bo
Source :
Journal of Medicinal Chemistry; 6/13/2024, Vol. 67 Issue 11, p8730-8756, 27p
Publication Year :
2024

Details

Language :
English
ISSN :
00222623
Volume :
67
Issue :
11
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
177895201
Full Text :
https://doi.org/10.1021/acs.jmedchem.4c00049