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Discovery of Covalent MLKL PROTAC Degraders via Optimization of a Theophylline Derivative Ligand for Treating Necroptosis.

Authors :
Li, Shang
Ma, Liangliang
Li, Xinxin
Jiang, Yuhan
Luo, Zhongwen
Yin, Fucheng
Zhang, Yonglei
Chen, Yifan
Wan, Siyuan
Zhou, Han
Kong, Lingyi
Wang, Xiaobing
Source :
Journal of Medicinal Chemistry; 9/12/2024, Vol. 67 Issue 17, p15353-15372, 20p
Publication Year :
2024

Details

Language :
English
ISSN :
00222623
Volume :
67
Issue :
17
Database :
Supplemental Index
Journal :
Journal of Medicinal Chemistry
Publication Type :
Academic Journal
Accession number :
179638757
Full Text :
https://doi.org/10.1021/acs.jmedchem.4c00949