Back to Search Start Over

7α-methoxy-2-[(substituted)methylene]cephem sulfones as inhibitors of human leukocyte elastase and thrombin

Authors :
Andhe V. Narender Reddy
David Czajkowski
Samarendra N. Maiti
Ronald G. Micetich
Charles Fiakpui
Jadwiga Kaleta
Source :
Chemistry of Heterocyclic Compounds. 34:1282-1288
Publication Year :
1998
Publisher :
Springer Science and Business Media LLC, 1998.

Abstract

A series of 7α-methoxy-2-[(substituted)methylene]cephem sulfones was synthesized. The compounds with an acetoxy group at the C-3′ position as a leaving group were found to be potent inhibitors of HLE. Selected compounds are also found to be antithrombin agents.

Details

ISSN :
15738353 and 00093122
Volume :
34
Database :
OpenAIRE
Journal :
Chemistry of Heterocyclic Compounds
Accession number :
edsair.doi...........5c621f29cf73b730efd66b989d53642e
Full Text :
https://doi.org/10.1007/bf02256808