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Simple Preparation ofN-Benzyl-β-aminohydroxamic Acidsby 1,3-Dipolar Cycloaddition­ of Nitrones

Authors :
Albert Defoin
Carine Chevrier
Source :
Synthesis. 2003:1221-1224
Publication Year :
2003
Publisher :
Georg Thieme Verlag KG, 2003.

Abstract

β-Aminohydroxamic acids 6a-d are prepared in 4 steps and 30-45% overall yield from nitrones la-d by 1,3-dipolar cycloaddition with phenyl vinyl ether, N-benzylation, thermal rearrangement, and nucleophilic substitution ofthe formed phenyl ester with hydroxylamine.

Details

ISSN :
1437210X and 00397881
Volume :
2003
Database :
OpenAIRE
Journal :
Synthesis
Accession number :
edsair.doi...........784840e3d174c8ee306860919615af02
Full Text :
https://doi.org/10.1055/s-2003-39412