Discovery of 2-(3-Benzamidopropanamido)thiazole-5-carboxylate Inhibitors of the Kinesin HSET (KIFC1) and the Development of Cellular Target Engagement Probes

Authors :: François Saint-Dizier
Thomas P. Matthews
Aaron M. Gregson
Hugues Prevet
Tatiana McHardy
Giampiero Colombano
Harry Saville
Martin Rowlands
Caroline Ewens
P. Craig McAndrew
Kathy Tomlin
Delphine Guillotin
Grace Wing-Yan Mak
Konstantinos Drosopoulos
Ioannis Poursaitidis
Rosemary Burke
Rob van Montfort
Spiros Linardopoulos
Ian Collins
Source :: Journal of Medicinal Chemistry. 66:2622-2645
Publication Year :: 2023
Publisher :: American Chemical Society (ACS), 2023.

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