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Metal-Free trans -Aziridination of Zerumbone: Synthesis and Biological Evaluation of Aziridine Derivatives of Zerumbone

Authors :
Kokkuvayil Vasu Radhakrishnan
P. Nisha
Jayaram Saranya
Thekke V. Baiju
Mangalam S. Nair
T. R. Reshmitha
Greeshma Gopalan
Murugan Thulasi Meenu
B. P. Dhanya
Source :
European Journal of Organic Chemistry. 2017:3072-3077
Publication Year :
2017
Publisher :
Wiley, 2017.

Abstract

Herein, we describe a metal-free, iodosobenzenediacetate mediated trans-aziridination of zerumbone by the direct use of sulphonamides. The preliminary in vitro-screening showed better anti-proliferative and anti-diabetic activity compared to parent compound zerumbone.

Details

ISSN :
1434193X
Volume :
2017
Database :
OpenAIRE
Journal :
European Journal of Organic Chemistry
Accession number :
edsair.doi...........a2e8e090dd16f572e21ff87f4e4327da
Full Text :
https://doi.org/10.1002/ejoc.201700410